[HTML][HTML] Directly compressed rosuvastatin calcium tablets that offer hydrotropic and micellar solubilization for improved dissolution rate and extent of drug release

S Butt, SMF Hasan, MM Hassan, KM Alkharfy… - Saudi Pharmaceutical …, 2019 - Elsevier
The objective was to use caffeine and Soluplus® to improve the dissolution rate and to
maintain a concentration of BCS Class II rosuvastatin calcium that exceeds its solubility …

Production of rosuvastatin calcium nanoparticles using gas antisolvent technique: Experimental and optimization

M Najafi, N Esfandiari, B Honarvar… - Periodica Polytechnica …, 2021 - pp.omikk.bme.hu
The activity of pharmaceutical substances crucially depends on the bioavailability of the
substances. The bioavailability of drugs in body and their rate of dissolution in the biological …

Solubility and thermodynamics of apremilast in different mono solvents: Determination, correlation and molecular interactions

F Shakeel, N Haq, FK Alanazi, IA Alsarra - International Journal of …, 2017 - Elsevier
The solubility data of recently launched poorly soluble antipsoriatic drug apremilast (APM) in
any mono solvent or cosolvent mixtures with respect to temperature are not available in …

Physicochemical characterization and pharmacokinetic evaluation of rosuvastatin calcium incorporated solid lipid nanoparticles

FNS Al-Heibshy, E Başaran, R Arslan, N Öztürk… - International journal of …, 2020 - Elsevier
Rosuvastatin calcium (RCa) is a very efficient antihyperlipidemic agent, however, being a
BCS class II drug, results in poor oral bioavailability. The present study focused on the …

Solubility of a poorly soluble immunosuppressant in different pure solvents: Measurement, correlation, thermodynamics and molecular interactions

MA Kalam, AA Khan, A Alshamsan, A Haque… - Journal of Molecular …, 2018 - Elsevier
The objective of this research work was to measure the solubility of mycophenolate mofetil
(MPM) in ten different pure solvents at temperatures T= 298.2 K to 318.2 K and pressure p …

Hybrid Self‐Assembled Gel Beads for Tuneable pH‐Controlled Rosuvastatin Delivery

CC Piras, AK Patterson… - Chemistry–A European …, 2021 - Wiley Online Library
This article describes the fabrication of new pH‐responsive hybrid gel beads combining the
polymer gelator calcium alginate with two different low‐molecular‐weight gelators (LMWGs) …

Solubility determination of raloxifene hydrochloride in ten pure solvents at various temperatures: Thermodynamics-based analysis and solute–solvent interactions

A Ahad, F Shakeel, OA Alfaifi, M Raish, A Ahmad… - International Journal of …, 2018 - Elsevier
The purpose of the present study was to determine the solubility of raloxifene hydrochloride
(RHCl) in ten solvents: water, ethanol, isopropyl alcohol (IPA), ethylene glycol (EG) …

Solubility measurement, thermodynamics and molecular interactions of flufenamic acid in different neat solvents

S Alshehri, F Shakeel - Journal of Molecular Liquids, 2017 - Elsevier
The solubility data of poorly soluble anti-inflammatory drug flufenamic acid (FFA) are scarce
in literature. Therefore, in the current study, the solubility of FFA in eleven different neat …

Strategic design and clinical evaluation of a fixed-dose combination tablet comprising valsartan, amlodipine, rosuvastatin and ezetimibe for patients with hypertension …

TK Kim, JE Lee, K Jeong, MJ Baek, D Kim… - Journal of …, 2024 - Springer
Purpose The objective of this study was to design a fixed-dose combination (FDC) tablet
with minimal interaction of valsartan, amlodipine, rosuvastatin and ezetimibe to improve …

The use of Calcium Phosphate-based starter pellets for the preparation of Sprinkle IR MUPS formulation of Rosuvastatin Calcium

K Cal, B Mikolaszek, T Hess, M Papaioannou, J Lenik… - Pharmaceuticals, 2023 - mdpi.com
Sprinkle formulations represent an interesting concept of medicinal products aimed at the
steadily growing population of patients suffering from swallowing difficulties (dysphagia). In …