Current trends in computer aided drug design and a highlight of drugs discovered via computational techniques: A review

VT Sabe, T Ntombela, LA Jhamba… - European Journal of …, 2021 - Elsevier
Computer-aided drug design (CADD) is one of the pivotal approaches to contemporary pre-
clinical drug discovery, and various computational techniques and software programs are …

The impact of molecular dynamics on drug design: applications for the characterization of ligand–macromolecule complexes

J Mortier, C Rakers, M Bermudez, MS Murgueitio… - Drug discovery today, 2015 - Elsevier
Highlights•Which molecular dynamics (MD) techniques are available for drug design?•How
is MD used to investigate ligand–macromolecule complexes?•How are MD studies applied …

Molecular docking, simulation and binding free energy analysis of small molecules as PfHT1 inhibitors

AJ Owoloye, FC Ligali, OA Enejoh, AZ Musa, O Aina… - PloS one, 2022 - journals.plos.org
Antimalarial drug resistance has thrown a spanner in the works of malaria elimination. New
drugs are required for ancillary support of existing malaria control efforts. Plasmodium …

In silico screening of hundred phytocompounds of ten medicinal plants as potential inhibitors of nucleocapsid phosphoprotein of COVID-19: an approach to prevent …

R Rolta, R Yadav, D Salaria, S Trivedi… - Journal of …, 2021 - Taylor & Francis
Currently, there is no specific treatment to cure COVID-19. Many medicinal plants have
antiviral, antioxidant, antibacterial, antifungal, anticancer, wound healing etc. Therefore, the …

New series of thiazole derivatives: synthesis, structural elucidation, antimicrobial activity, molecular modeling and MOE docking

I Althagafi, N El-Metwaly, TA Farghaly - Molecules, 2019 - mdpi.com
Based on the extensive biological activities of thiazole derivatives against different types of
diseases, we are interested in the effective part of many natural compounds, so we …

Identification of 1H-purine-2, 6-dione derivative as a potential SARS-CoV-2 main protease inhibitor: molecular docking, dynamic simulations, and energy calculations

H Nada, A Elkamhawy, K Lee - PeerJ, 2022 - peerj.com
The rapid spread of the coronavirus since its first appearance in 2019 has taken the world by
surprise, challenging the global economy, and putting pressure on healthcare systems …

Computational identification of potential inhibitors targeting cdk1 in colorectal cancer

UC Ogbodo, OA Enejoh, CH Okonkwo… - Frontiers in …, 2023 - frontiersin.org
Introduction: Despite improved treatment options, colorectal cancer (CRC) remains a huge
public health concern with a significant impact on affected individuals. Cell cycle …

Design, synthesis, molecular docking studies and biological evaluation of thiazole carboxamide derivatives as COX inhibitors

M Hawash, N Jaradat, M Abualhasan, MK Şüküroğlu… - BMC chemistry, 2023 - Springer
Background Nonsteroidal anti-inflammatory drugs (NSAIDs) have been the most commonly
used class of medications worldwide for the last three decades. Objectives This study aimed …

Insight into antioxidant-like activity and computational exploration of identified bioactive compounds in Talinum triangulare (Jacq.) aqueous extract as potential …

OB Afolabi, OR Olasehinde, OV Owolabi… - … Medicine and Therapies, 2024 - Springer
Background Recent reports have highlighted the significance of plant bioactive components
in drug development targeting neurodegenerative disorders such as Alzheimer's disease …

[HTML][HTML] High-throughput screening and molecular dynamics simulation of natural product-like compounds against Alzheimer's disease through multitarget approach

D Iqbal, MT Rehman, A Bin Dukhyil, SMD Rizvi… - Pharmaceuticals, 2021 - mdpi.com
Alzheimer's disease (AD) is a progressive neurological disorder that affects 50 million
people. Despite this, only two classes of medication have been approved by the FDA …