The evolving small‐molecule fluorescent‐conjugate toolbox for C lass A GPCRs

AJ Vernall, SJ Hill, B Kellam - British journal of pharmacology, 2014 - Wiley Online Library
The past decade has witnessed fluorescently tagged drug molecules gaining significant
attraction in their use as pharmacological tools with which to visualize and interrogate …

Biomarker-targeted fluorescent probes for breast cancer imaging

D Yue, M Wang, F Deng, W Yin, H Zhao, X Zhao… - Chinese Chemical …, 2018 - Elsevier
Breast cancer has become a common tumor worldwide which seriously endangers people's
health. Early diagnosis and treatment are particularly urgent in order to reduce the onset …

Detection of an estrogen derivative in two breast cancer cell lines using a single core multimodal probe for imaging (SCoMPI) imaged by a panel of luminescent and …

S Clede, F Lambert, C Sandt, S Kascakova, M Unger… - Analyst, 2013 - pubs.rsc.org
3-Methoxy-17α-ethynylestradiol or mestranol is a prodrug for ethynylestradiol and the
estrogen component of some oral contraceptive formulations. We demonstrate here that a …

Correlating molecular character of NIR imaging agents with tissue-specific uptake

EA Owens, H Hyun, JG Tawney, HS Choi… - Journal of medicinal …, 2015 - ACS Publications
Near-infrared (NIR) fluorescent contrast agents are emerging in optical imaging as sensitive,
cost-effective, and nonharmful alternatives to current agents that emit harmful ionizing …

Molecular fluorescence, phosphorescence, and chemiluminescence spectrometry

S Das, AM Powe, GA Baker, B Valle… - Analytical …, 2012 - ACS Publications
As a result of change in due date, this Review covers the one and two-third-year period
since our last review1 from January 2010 through August 2011. Manuscripts outside this …

Recent advances in receptor-targeted fluorescent probes for in vivo cancer imaging

M Bai, DJ Bornhop - Current medicinal chemistry, 2012 - ingentaconnect.com
Receptor-targeted optical imaging of cancer is emerging as an attractive strategy for early
cancer diagnosis and surgical guidance. The success of such strategy depends largely …

Review of fluorescent steroidal ligands for the estrogen receptor 1995–2018

N Gajadeera, RN Hanson - Steroids, 2019 - Elsevier
The development of fluorescent ligands for the estrogen receptor (ER) continues to be of
interest. Over the past 20 years, most efforts have focused on appending an expanding …

Near infrared molecular imaging of breast cancer cell lines using a novel ER targeted fluorescent dye

VJ Pillai, I Jose - 2022 - researchsquare.com
Hormone-targeted contrast agents bind with functional groups associated with the
physiology of breast cancer leading to improved prognosis. We have synthesized a novel …

Cell-selective breast cancer targeting through estrogen receptors

BD Kurmi, R Paliwal, SR Paliwal - Targeted Nanomedicine for Breast …, 2022 - Elsevier
Breast cancer is the foremost cause of death among women worldwide. The estrogen
receptors (ERs), a nuclear receptor superfamily member, are closely associated with breast …

Emerging Technologies in Breast Imaging

MS Newell, AI Holbrook - Breast Cancer Screening and Diagnosis: A …, 2014 - Springer
Mammographic screening has been validated as an effective way to decrease breast cancer
deaths, responsible for a 30–40% mortality reduction in participating populations. However …