Estrogen receptor function: impact on the human endometrium

K Yu, ZY Huang, XL Xu, J Li, XW Fu… - Frontiers in …, 2022‏ - frontiersin.org
The physiological role of estrogen in the female endometrium is well established. On the
basis of responses to steroid hormones (progesterone, androgen, and estrogen), the …

Estrogen receptor signaling in the immune system

B Chakraborty, J Byemerwa, T Krebs, F Lim… - Endocrine …, 2023‏ - academic.oup.com
The immune system functions in a sexually dimorphic manner, with females exhibiting more
robust immune responses than males. However, how female sex hormones affect immune …

The Concise Guide to PHARMACOLOGY 2013/14: G protein‐coupled receptors

SPH Alexander, HE Benson… - British journal of …, 2013‏ - Wiley Online Library
Abstract The Concise Guide to PHARMACOLOGY 2013/14 provides concise overviews of
the key properties of over 2000 human drug targets with their pharmacology, plus links to an …

Twenty years of the G protein-coupled estrogen receptor GPER: Historical and personal perspectives

M Barton, EJ Filardo, SJ Lolait, P Thomas… - The Journal of steroid …, 2018‏ - Elsevier
Estrogens play a critical role in many aspects of physiology, particularly female reproductive
function, but also in pathophysiology, and are associated with protection from numerous …

Does GPER Really Function as a G Protein-Coupled Estrogen Receptor in vivo?

J Luo, D Liu - Frontiers in endocrinology, 2020‏ - frontiersin.org
Estrogen can elicit pleiotropic cellular responses via a diversity of estrogen receptors (ERs)—
mediated genomic and rapid non-genomic mechanisms. Unlike the genomic responses …

Birth and death of bone cells: basic regulatory mechanisms and implications for the pathogenesis and treatment of osteoporosis

SC Manolagas - Endocrine reviews, 2000‏ - academic.oup.com
The adult skeleton regenerates by temporary cellular structures that comprise teams of
juxtaposed osteoclasts and osteoblasts and replace periodically old bone with new. A …

Estrogen carcinogenesis in breast cancer

JD Yager, NE Davidson - New England Journal of Medicine, 2006‏ - Mass Medical Soc
Estrogen Carcinogenesis in Breast Cancer | New England Journal of Medicine Skip to main
content The New England Journal of Medicine homepage Advanced Search SEARCH …

Mechanisms of estrogen receptor signaling: convergence of genomic and nongenomic actions on target genes

L Björnström, M Sjöberg - Molecular endocrinology, 2005‏ - academic.oup.com
Estrogen receptors (ERs) act by regulating transcriptional processes. The classical
mechanism of ER action involves estrogen binding to receptors in the nucleus, after which …

Estrogen-Induced Activation of Erk-1 and Erk-2 Requires the G Protein-Coupled Receptor Homolog, GPR30, and Occurs via Trans-Activation of the Epidermal Growth …

EJ Filardo, JA Quinn, KI Bland… - Molecular …, 2000‏ - academic.oup.com
Estrogen rapidly activates the mitogen-activated protein kinases, Erk-1 and Erk-2, via an as
yet unknown mechanism. Here, evidence is provided that estrogen-induced Erk-1/-2 …

Estrogen receptor null mice: what have we learned and where will they lead us?

JF Couse, KS Korach - Endocrine reviews, 1999‏ - academic.oup.com
Elwood Jensen and Jack Gorski had spent 10 yr providing experimental evidence to support
the concept of an intracellular “receptor” protein for steroid hormones. Their combined work …