In silico pharmacology for drug discovery: methods for virtual ligand screening and profiling

S Ekins, J Mestres, B Testa - British journal of pharmacology, 2007 - Wiley Online Library
Pharmacology over the past 100 years has had a rich tradition of scientists with the ability to
form qualitative or semi‐quantitative relations between molecular structure and activity in …

Homology modeling in drug discovery: current trends and applications

CN Cavasotto, SS Phatak - Drug discovery today, 2009 - Elsevier
As structural genomics (SG) projects continue to deposit representative 3D structures of
proteins, homology modeling methods will play an increasing role in structure-based drug …

Structure-based prediction of protein–protein interactions on a genome-wide scale

QC Zhang, D Petrey, L Deng, L Qiang, Y Shi, CA Thu… - Nature, 2012 - nature.com
The genome-wide identification of pairs of interacting proteins is an important step in the
elucidation of cell regulatory mechanisms,. Much of our present knowledge derives from …

Comparative protein structure modeling using MODELLER

B Webb, A Sali - Current protocols in bioinformatics, 2016 - Wiley Online Library
Comparative protein structure modeling predicts the three‐dimensional structure of a given
protein sequence (target) based primarily on its alignment to one or more proteins of known …

Statistical potential for assessment and prediction of protein structures

M Shen, A Sali - Protein science, 2006 - Wiley Online Library
Protein structures in the Protein Data Bank provide a wealth of data about the interactions
that determine the native states of proteins. Using the probability theory, we derive an atomic …

The SWISS-MODEL Repository and associated resources

F Kiefer, K Arnold, M Künzli, L Bordoli… - Nucleic acids …, 2009 - academic.oup.com
Abstract SWISS-MODEL Repository (http://swissmodel. expasy. org/repository/) is a
database of 3D protein structure models generated by the SWISS-MODEL homology …

[HTML][HTML] Population genomics reveal recent speciation and rapid evolutionary adaptation in polar bears

S Liu, ED Lorenzen, M Fumagalli, B Li, K Harris… - Cell, 2014 - cell.com
Polar bears are uniquely adapted to life in the High Arctic and have undergone drastic
physiological changes in response to Arctic climates and a hyperlipid diet of primarily …

Protein structure modeling with MODELLER

N Eswar, D Eramian, B Webb, MY Shen… - Structural proteomics: high …, 2008 - Springer
Genome sequencing projects have resulted in a rapid increase in the number of known
protein sequences. In contrast, only about one-hundredth of these sequences have been …

ModBase, a database of annotated comparative protein structure models and associated resources

U Pieper, BM Webb, GQ Dong… - Nucleic acids …, 2014 - academic.oup.com
Abstract ModBase (http://salilab. org/modbase) is a database of annotated comparative
protein structure models. The models are calculated by ModPipe, an automated modeling …

Progress and challenges in protein structure prediction

Y Zhang - Current opinion in structural biology, 2008 - Elsevier
Depending on whether similar structures are found in the PDB library, the protein structure
prediction can be categorized into template-based modeling and free modeling. Although …