Extending the potency and lifespan of antibiotics: inhibitors of gram-negative bacterial efflux pumps

M Duffey, RP Jumde, RMA da Costa… - ACS Infectious …, 2024 - ACS Publications
Efflux is a natural process found in all prokaryotic and eukaryotic cells that removes a
diverse range of substrates from inside to outside. Many antibiotics are substrates of …

[PDF][PDF] Design, synthesis and bioactivity studies of novel triazolopyrimidinone compounds

H Istanbullu, G Bayraktar, I Ozturk, R Coban… - J Res Pharm, 2022 - jrespharm.com
This study was aimed to develop novel compounds to combat antimicrobial resistance,
which is one of the biggest threats to global health. For this purpose, compounds bearing …