The assembly of architecturally complex alkaloids embedding the indole nucleus is of
paramount importance for the target oriented synthesis of biologically active molecules. 1 A …

The first catalytic asymmetric construction of 3, 3′‐bisindole skeletons bearing both axial
and central chirality has been established by organocatalytic asymmetric addition reactions …

The indole 3-position is highly electron-rich and typically functions as the primary
nucleophilic site to react with a large array of electrophiles, leading to various functionalized …

The electrophilic intermediate, vinylogous imine or vinylogous iminium, can be in situ
generated from 3-indolyl-methanols under acidic conditions. With the aid of chiral catalysts …

A catalytic asymmetric synthesis of 3, 3′-bisindoles bearing single axial chirality has been
established via chiral phosphoric acid (CPA)-catalyzed enantioselective addition reaction of …

A copper-catalyzed Friedel–Crafts propargylation/hydroamination/aromatization sequence
is described. In the presence of a catalytic amount of CuI, this sequential reaction can …

A palladium catalyzed, carbon monoxide mediated, double reductive cyclization of 1, 4-, 1, 3-
, and 2, 3-bis (2-nitroaryl)-1, 3-butadienes to afford 2, 2′-, 2, 3′-, and 3, 3′-biindoles …

A method for the rapid synthesis of polycyclic 3, 3′-biindole derivatives has been
developed through AgOTf-catalyzed nucleophilic addition and cycloisomerization …

Abstract The Masuda borylation/Suzuki arylation (MBSA) sequence starting from N‐
protected 3‐iodoindoles has successfully been extended to the coupling of five‐membered …

A simple route for the synthesis of 1, 4-benzoxazin-3-(4H)-ones is described herein. This
method involves the reductive cyclization of 2-(2-nitrophenoxy) acetonitrile adducts in the …