Oxidative coupling with S–N bond formation

OM Mulina, AI Ilovaisky… - European Journal of …, 2018 - Wiley Online Library
Oxidative strategies are a powerful tool in organic synthesis for the formation of heteroatom–
heteroatom, carbon–heteroatom, and carbon–carbon bonds. Among these processes the …

Progress in copper-catalysed/mediated intramolecular dehydrogenative coupling

RP Bhaskaran, KH Nayak, MK Sreelekha… - Organic & Biomolecular …, 2023 - pubs.rsc.org
Transition metal-catalysed C–H functionalization reactions are one of the most efficient
synthetic methodologies to construct carbon–carbon and carbon–heteroatom bonds. The …

Design and synthesis of thiourea-based derivatives as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors

ŞD Doğan, MG Gündüz, H Doğan, VS Krishna… - European journal of …, 2020 - Elsevier
Tuberculosis remains the most deadly infectious disease worldwide due to the emergence
of drug-resistant strains of Mycobacterium tuberculosis. Hence, there is a great need for …

Discovery of hydrazone containing thiadiazoles as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors

H Doğan, ŞD Doğan, MG Gündüz, VS Krishna… - European Journal of …, 2020 - Elsevier
Tuberculosis, caused by Mycobacterium tuberculosis, is a serious infectious disease and
remains a global health problem. There is an increasing need for the discovery of novel …

Acyl azides: Versatile compounds in the synthesis of various heterocycles

M Balci - Synthesis, 2018 - thieme-connect.com
Carbon–nitrogen bond formation is one of the most important reactions in organic chemistry.
Various synthetic strategies for the generation of C–N bonds are described in the literature …

1, 3-Disubstituted urea derivatives: Synthesis, antimicrobial activity evaluation and in silico studies

MG Gündüz, SB Uğur, F Güney, C Özkul, VS Krishna… - Bioorganic …, 2020 - Elsevier
The development of new antimicrobial compounds is in high demand to overcome the
emerging drug resistance against infectious microbial pathogens. In the present study, we …

Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities

R Keleş Atıcı, ŞD Doğan, MG Gündüz… - Drug Development …, 2022 - Wiley Online Library
The recent emergence of drug‐resistant strains of Mycobacterium tuberculosis (Mtb) has
complicated and significantly slowed efforts to eradicate and/or reduce the worldwide …

Chemodivergent Synthesis of Benzothiadiazin-3-one 1-Oxides and Benzisothiazol-3-ones via Visible Light-Promoted Intramolecular N–S Bond Formation

H Li, Z **ong, S Sheng, J Chen - The Journal of Organic …, 2023 - ACS Publications
We reported a versatile protocol to chemodivergently construct significant heterocyclic
scaffolds of benzothiadiazin-3-one 1-oxides and benzisothiazol-3-ones by visible light …