A review of the biological activities of heterocyclic compounds comprising oxadiazole moieties

BF Ruan, QL Guo, QS Li, LZ Li… - Current Topics in …, 2022 - ingentaconnect.com
The oxadiazole core is considered a privileged moiety in many medicinal chemistry
applications. The oxadiazole class includes 1, 2, 3-oxadiazole, 1, 2, 4-oxadiazole, 1, 3, 4 …

New quinoxaline-oxadiazole hybrids as tubulin inhibitors: Synthesis, cytotoxicity, and molecular dynamics simulations

BR Vancha, M Sreeshitha, KP Vasikarla… - Journal of Molecular …, 2025 - Elsevier
This study describes the synthesis and biological evaluation of a series of novel quinoxaline-
oxadiazole hybrid compounds. These compounds were designed to enhance anticancer …

Oxadiazoles have butyrate-specific conditional activity against Mycobacterium tuberculosis

JV Early, A Casey, MA Martinez-Grau… - Antimicrobial agents …, 2016 - Am Soc Microbiol
Mycobacterium tuberculosis is a global pathogen of huge importance which can adapt to
several host niche environments in which carbon source availability is likely to vary. We …

Synthesis and electrochemical and antioxidant properties of chalcogenocyanate oxadiazole and 5-heteroarylchalcogenomethyl-1 H-tetrazole derivatives

JG Leal, AC Sauer, JCP Mayer, ST Stefanello… - New Journal of …, 2017 - pubs.rsc.org
This article presents the chalcogenocyanate oxadiazoles 7 and 8 and their derivatives 5-
heteroarylchalcogenomethyl-1H-tetrazoles 9 and 10, which were synthesized in high yields …

[PDF][PDF] Synthesis & characterization of some 1, 3, 4-oxadiazolederivatives & new cyclic imides from creatinine

MI Kalaf, OS Hashim - Iraqi Journal of Science, 2015 - iasj.net
Abstract A series of new 1, 3, 4-oxadiazole derivatives and cyclic Imides containing
Creatinine heterocyclic molecule were prepared via following method: first step included …

Síntese e caracterização dos 3-(benzo [c][1, 2, 5] calcogenodiazol-5-il)-5-(ariletinil) 1, 2, 4-oxadiazóis derivados de (z)-n'-hidroxibenzo [c][1, 2, 5] calcogenodiazóis-5 …

PC Pereira - 2023 - repositorio.ufsm.br
The importance of heterocycle chemistry has grown in recent years, enabling the connection
among many interdisciplinary areas of science, standing out in synthetic organic chemistry …

Synthesis and Biological Evaluation of 2-methoxy-N-phenyl-6-(5-phenyl-1, 3, 4-oxadiazol-2-yl) pyridin-3-amine Derivatives as Antimicrobial Agents

V Namani, B Bharath Kumar Goud… - Letters in Organic …, 2016 - ingentaconnect.com
Background: A series of novel 2-methoxy-N-phenyl-6-(5-phenyl-1, 3, 4-oxadiazol-2-yl)
pyridin-3-amine (6a-i) have been synthesized from bromo methoxy picolinicacid as starting …

[HTML][HTML] 5-(4-Methylphenyl)-1, 3, 4-oxadiazol-2-amine

J Zheng, W Li, M Song, Y Xu - Acta Crystallographica Section E …, 2012 - scripts.iucr.org
organic compounds Page 1 5-(4-Methylphenyl)-1,3,4-oxadiazol-2amine Juan Zheng, Wen-juan
Li, Manman Song and Yan Xu* Department of Chemistry, Zhengzhou University, Zhengzhou …

[PDF][PDF] INTERNATIONAL RESEARCH JOURNAL OF PHARMACY

NTOE BIOAVAILABILITY - academia.edu
Oral route is the most important and preferred route for drug administration due to the
convenience, ease of administration and patient compliance. Tablet is the most preferred …

[ZITATION][C] short review on 1, 3, 4–oxadiazole and its pharmacological activities

AS D'souza, A D'Souza, AP Mendonca, BA Noronha - J. **an Shiyou Uni