[HTML][HTML] Natural and bioinspired excipients for dry powder inhalation formulations

D Zillen, M Beugeling, WLJ Hinrichs, HW Frijlink… - Current Opinion in …, 2021‏ - Elsevier
Pulmonary drug delivery can have several advantages over other administration routes, in
particular when using dry powder formulations. Such dry powder inhalation formulations …

Excipients for Novel Inhaled Dosage Forms: An Overview

C Yousry, M Goyal, V Gupta - AAPS PharmSciTech, 2024‏ - Springer
Pulmonary drug delivery is a form of local targeting to the lungs in patients with respiratory
disorders like cystic fibrosis, pulmonary arterial hypertension (PAH), asthma, chronic …

Inhaled deep eutectic solvent based-nanoemulsion of pirfenidone in idiopathic pulmonary fibrosis

JH Kang, MS Yang, TK Kwon, DW Kim… - Journal of Controlled …, 2022‏ - Elsevier
Pirfenidone (PRF), the first FDA-approved drug to treat idiopathic pulmonary fibrosis (IPF)
and formulated as an oral dosage form, has many side effects. To enhance the therapeutic …

Preparation of orodispersible tablets of bosentan using xylitol and menthol as dissolution enhancers

RM Sakr, AES Abdelaziz, EA Mazyed… - Scientific Reports, 2024‏ - nature.com
Bosentan is a drug used to treat pulmonary hypertension via dual endothelial receptor
antagonism. Bosentan has a restricted oral bioavailability, a problem that's mostly due to …

Customizable resveratrol spray-dried micro-composites for inhalation as a promising contender for treatment of idiopathic pulmonary fibrosis

S Ahmed, M Mansour, RAH Ishak… - International Journal of …, 2023‏ - Elsevier
The past decades have witnessed tremendous expansion in utilization of plant-derived
medicines as resveratrol (RES) in treating several diseases like idiopathic pulmonary …

In vivo pharmacokinetic and pharmacodynamic study of inhalable pirfenidone microparticles prepared via high-energy bead milling

JH Kang, JC Choi, WY Song, J Choi, SH Lee… - Journal of …, 2023‏ - Springer
Purpose Pirfenidone (PRF) is the first FDA-approved active pharmaceutical ingredient for
the treatment of idiopathic pulmonary fibrosis (IPF). However, it has severe adverse effects …

[HTML][HTML] Preparation and in vivo evaluation of a lidocaine self-nanoemulsifying ointment with glycerol monostearate for local delivery

JH Kang, KH Yoo, HY Park, SM Hyun, SD Han… - Pharmaceutics, 2021‏ - mdpi.com
Lidocaine, a commonly used local anesthetic, has recently been developed into a number of
ointment products to treat hemorrhoids. This study examined its efficient delivery to the …

Development of spray-dried N-acetylcysteine dry powder for inhalation

L Mancini, M Paolantoni, A Schoubben… - International Journal of …, 2023‏ - Elsevier
N-acetylcysteine (NAC) has both antioxidant and immunomodulatory activities and has been
used as adjuvant therapy in several viral infections. Recently, NAC attracted attention for its …

High energy ball milling vs. nano spray drying in the development of supersaturated systems loaded with bosentan

A Krupa, F Danede, D Majda, A Węgrzyn… - European Journal of …, 2023‏ - Elsevier
In this study, high energy ball milling and nano spray drying were used to prepare
amorphous solid dispersions of bosentan in copovidone for the first time. In particular, the …

[HTML][HTML] Co-spray dried nafamostat mesylate with lecithin and mannitol as respirable microparticles for targeted pulmonary delivery: pharmacokinetics and lung …

JH Kang, YJ Kim, MS Yang, DH Shin, DW Kim, IY Park… - Pharmaceutics, 2021‏ - mdpi.com
Coronavirus disease 2019 (COVID-19), caused by a new strain of coronavirus called severe
acute respiratory syndrome coronavirus 2 (SARS-CoV-2), is spreading rapidly worldwide …