Acetamides: chemotherapeutic agents for inflammation-associated cancers
Now clear evidences are available to support the hypothesis that inflammation accelerates
the conditions including events and molecules that reach to various types of cancers …
the conditions including events and molecules that reach to various types of cancers …
Novel 1, 2, 4‐triazole derivatives: Design, synthesis, anticancer evaluation, molecular docking, and pharmacokinetic profiling studies
Abstract Three novel series of 1, 2, 4‐triazole derivatives were designed and synthesized as
potential adenosine A2B receptor antagonists. The design of the new compounds depended …
potential adenosine A2B receptor antagonists. The design of the new compounds depended …
[HTML][HTML] N-Phenyl-2-p-tolylthiazole-4-carboxamide derivatives: Synthesis and cytotoxicity evaluation as anticancer agents
Objective (s): According to the prevalence of neoplastic diseases, there is a deep necessity
for discovery of novel anticancer drugs in the field of medicinal chemistry. In the current …
for discovery of novel anticancer drugs in the field of medicinal chemistry. In the current …
[HTML][HTML] N-(5-Mercapto-1, 3, 4-thiadiazol-2-yl)-2-phenylacetamide derivatives: synthesis and in-vitro cytotoxicity evaluation as potential anticancer agents
A Mohammadi-Farani, N Heidarian… - Iranian Journal of …, 2014 - ncbi.nlm.nih.gov
A new series of N-(5-Mercapto-1, 3, 4-thiadiazol-2-yl)-2-phenylacetamide derivatives (3a-3j)
were synthesized via an amidation reaction using EDC and HOBt in acetonitrile solvent at …
were synthesized via an amidation reaction using EDC and HOBt in acetonitrile solvent at …
Synthesis and evaluation of anticonvulsant activity of (Z)-4-(2-oxoindolin-3-ylideneamino)-N-phenylbenzamide derivatives in mice
Due to resistance of some epileptic patients to the current medications and the general
incidence of severe side effects of these drugs, development and discovery of novel …
incidence of severe side effects of these drugs, development and discovery of novel …
Phytoconstituents from Curcuma longa L. aqueous ethanol extract and its immunomodulatory effect on diabetic infected rats
MH Shabana, EM Shahy, MM Taha… - Egyptian …, 2015 - journals.lww.com
Materials and methods The extraction and isolation of the constituents of C. longa were
performed according to the standard methods of column, paper, and thin-layer …
performed according to the standard methods of column, paper, and thin-layer …
Biophysical investigation and antitumor potential of heterocyclic palladium-based agent: cytotoxicity, spectroscopic and molecular docking approaches in interaction …
M Saeidifar, R Sabbaghzadeh… - Polycyclic Aromatic …, 2021 - Taylor & Francis
With the aim of cancer treatment, interaction between 1-hexyldithiocarbamato 1, 10-
phenanthrolinepalladium (II) nitrate complex ([Pd (Hex-Dtc)(Phen)] NO3, Pd-HDP), as a …
phenanthrolinepalladium (II) nitrate complex ([Pd (Hex-Dtc)(Phen)] NO3, Pd-HDP), as a …
[HTML][HTML] Synthesis and Biological Evaluation of N-(5-(pyridin-2-yl)-1, 3, 4-thiadiazol-2-yl) benzamide Derivatives as Lipoxygenase Inhibitor with Potential Anticancer …
In the recent years, the role of LOX enzymes in the origin of neoplastic diseases such as
colorectal, skin, pancreatic and renal cancers has been confirmed. A new series of 1, 3, 4 …
colorectal, skin, pancreatic and renal cancers has been confirmed. A new series of 1, 3, 4 …
[PDF][PDF] 4-Halo-N-(5-(trifluoromethyl)-1, 3, 4-thiadiazol-2-yl) benzamide and Benzothioamide Derivatives: Synthesis and in vitro Anticancer Assessment
AR Aliabadi, H Harasami Neek, Y Bahmani - Iranian Journal of Chemistry …, 2020 - ijcce.ac.ir
Cancer is a lethal disorder that has caused a serious threat to human health and nowadays
there is a crucial need for the development of novel anticancer agents. A new series of 1, 3 …
there is a crucial need for the development of novel anticancer agents. A new series of 1, 3 …
Synthesis and acetylcholinesterase inhibitory assessment of benzamide derivatives incorporated piperazine moiety as potential anti-Alzheimer agents
According to the obtained information from X-ray crystallography, it has been characterized
that two distinct parts are observable in the active site of AChE.[...] the ethylacetate was …
that two distinct parts are observable in the active site of AChE.[...] the ethylacetate was …