[HTML][HTML] A comprehensive review on pyrazoline based heterocyclic hybrids as potent anticancer agents

K Haider, M Shafeeque, S Yahya, MS Yar - European Journal of Medicinal …, 2022 - Elsevier
Cancer is one of the leading causes of death globally, around 10 million deaths are reported
every year due to cancer. Some clinically approved anticancer drugs play a riveting role in …

[HTML][HTML] Pyrazoline hybrids as promising anticancer agents: An up-to-date overview

D Matiadis, M Sagnou - International Journal of Molecular Sciences, 2020 - mdpi.com
Pyrazolines are five-membered heterocycles possessing two adjacent nitrogens. They have
attracted significant attention from organic and medicinal chemists due to their potent …

Thiazole derivatives in medicinal chemistry: Recent advancements in synthetic strategies, structure activity relationship and pharmacological outcomes

A Singh, D Malhotra, K Singh, R Chadha… - Journal of Molecular …, 2022 - Elsevier
Thiazole derivatives remains honored heterocycles in the field of medicinal chemistry. This
scaffold has been proven as a universal motif that is present in numerous pharmacologically …

Novel metabolic enzyme inhibitors designed through the molecular hybridization of thiazole and pyrazoline scaffolds

B Sever, C Türkeş, MD Altıntop, Y Demir… - Archiv der …, 2021 - Wiley Online Library
New hybrid thiazolyl–pyrazoline derivatives (4a–k) were obtained through a facile and
versatile synthetic procedure, and their inhibitory effects on the human carbonic anhydrase …

[HTML][HTML] 1, 3, 4-Oxadiazole-containing hybrids as potential anticancer agents: Recent developments, mechanism of action and structure-activity relationships

S Nayak, SL Gaonkar, EA Musad… - Journal of Saudi Chemical …, 2021 - Elsevier
Chemotherapy is an important therapeutic approach for the treatment of cancer. Currently,
many anticancer drugs are available in the market that plays an important role in cancer …

Thiazolyl-pyrazoline derivatives: In vitro and in silico evaluation as potential acetylcholinesterase and carbonic anhydrase inhibitors

B Sever, C Türkeş, MD Altıntop, Y Demir… - International Journal of …, 2020 - Elsevier
Alzheimer's disease (AD) is a complex, predominant, and progressive form of dementia. The
treatment of AD alters depending on the cognitive and behavioral symptoms. The utility of …

Development in the synthesis of bioactive thiazole-based heterocyclic hybrids utilizing phenacyl bromide

G Kumari, S Dhillon, P Rani, M Chahal, DK Aneja… - ACS …, 2024 - ACS Publications
Heterocyclic hybrid frameworks represent a burgeoning domain within the realms of drug
discovery and medicinal chemistry, attracting considerable attention in recent years …

New pyrazolyl-thiazolidinone/thiazole derivatives as celecoxib/dasatinib analogues with selective COX-2, HER-2 and EGFR inhibitory effects: design, synthesis, anti …

WAA Fadaly, TH Zidan, NM Kahk… - Journal of enzyme …, 2023 - Taylor & Francis
Two new series of pyrazolyl-thiazolidinone/thiazole derivatives 16a–b and 18a–j were
synthesised, merging the scaffolds of celecoxib and dasatinib. Compounds 16a, 16b and 18f …

A comprehensive review on thiazole based conjugates as anti-cancer agents

R Rana, N Kumar, HK Gulati, A Sharma… - Journal of Molecular …, 2023 - Elsevier
Over the past few decades, a significant number of anticancer drugs have been developed,
both natural and synthetic. Thiazole, a 5-membered distinctive heterocyclic motif with …

[HTML][HTML] New Thiazolyl-Pyrazoline derivatives as potential dual EGFR/HER2 inhibitors: design, synthesis, anticancer activity evaluation and in silico study

MM Fakhry, AA Mattar, M Alsulaimany, EM Al-Olayan… - Molecules, 2023 - mdpi.com
A new series of thiazolyl-pyrazoline derivatives (4a–d, 5a–d 6a, b, 7a–d, 8a, b, and 10a, b)
have been designed and synthesized through the combination of thiazole and pyrazoline …