Strategies to address low drug solubility in discovery and development

HD Williams, NL Trevaskis, SA Charman… - Pharmacological …, 2013‏ - Elsevier
Drugs with low water solubility are predisposed to low and variable oral bioavailability and,
therefore, to variability in clinical response. Despite significant efforts to “design in” …

Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates

N Blagden, M de Matas, PT Gavan, P York - Advanced drug delivery …, 2007‏ - Elsevier
The increasing prevalence of poorly soluble drugs in development provides notable risk of
new products demonstrating low and erratic bioavailabilty with consequences for safety and …

Compression physics in the formulation development of tablets

S Patel, AM Kaushal, AK Bansal - Critical Reviews™ in …, 2006‏ - dl.begellhouse.com
The advantages of high-precision dosing, manufacturing efficiency, and patient compliance
make tablets the most popular dosage forms. Compaction, an essential manufacturing step …

Phase transition enthalpy measurements of organic and organometallic compounds and ionic liquids. Sublimation, vaporization, and fusion enthalpies from 1880 to …

W Acree, JS Chickos - Journal of Physical and Chemical Reference …, 2017‏ - pubs.aip.org
The second part of this compendium concludes with a collection of phase change enthalpies
of organic molecules inclusive of C 11–C 192 reported over the period 1880–2015. Also …

Drug carrier systems for solubility enhancement of BCS class II drugs: a critical review

S Kumar, D Bhargava, A Thakkar… - Critical Reviews™ in …, 2013‏ - dl.begellhouse.com
Poor aqueous solubility impedes a drug's bioavailability and challenges its pharmaceutical
development. Pharmaceutical development of drugs with poor water solubility requires the …

Formation of phenytoin nanoparticles using rapid expansion of supercritical solution with solid cosolvent (RESS-SC) process

R Thakur, RB Gupta - International journal of pharmaceutics, 2006‏ - Elsevier
Nanoparticles are of significant importance in drug delivery. Rapid expansion of supercritical
solution (RESS) process can produce pure and high-quality drug particles. However, due to …

Process intensification for pharmaceutical crystallization

J Wang, F Li, R Lakerveld - Chemical Engineering and Processing-Process …, 2018‏ - Elsevier
Process intensification (PI) provides great opportunities to drastically improve the
performance of chemical processes within many branches of chemical industry including the …

Multistage crystallization of plate-like crystals: A modeling and experimental study on adipic acid

D Biri, A Jaeggi, P Malach, AK Rajagopalan… - Crystal Growth & …, 2024‏ - ACS Publications
Particles exhibiting a plate-like shape, encountered during crystallization, present
challenges in downstream processing. Consequently, it is crucial to manipulate the size and …

Impact of crystal habit on biopharmaceutical performance of celecoxib

SR Modi, AKR Dantuluri, V Puri, YB Pawar… - Crystal growth & …, 2013‏ - ACS Publications
Poor biopharmaceutical performance of Biopharmaceutical Classification System (BCS)
class II drug molecules is a major hurdle in the design and development of pharmaceutical …

Nano-extrusion: A promising tool for continuous manufacturing of solid nano-formulations

R Baumgartner, A Eitzlmayr, N Matsko… - International journal of …, 2014‏ - Elsevier
Since more than 40% of today's drugs have low stability, poor solubility and/or limited ability
to cross certain biological barriers, new platform technologies are required to address these …