Recent developments and biological activities of thiazolidinone derivatives: A review
Thiazolidinone is considered as a biologically important active scaffold that possesses
almost all types of biological activities. Successful introduction of ralitoline as a potent anti …
almost all types of biological activities. Successful introduction of ralitoline as a potent anti …
4-Thiazolidinones: the advances continue…
The diversity in the biological response of 4-thiazolidinones has attracted the attention of
many researchers to explore this framework for its potential. It is, therefore, of prime …
many researchers to explore this framework for its potential. It is, therefore, of prime …
Synthetic approaches, structure activity relationship and biological applications for pharmacologically attractive pyrazole/pyrazoline–thiazolidine-based hybrids
The features of the chemistry of 4-thiazolidinone and pyrazole/pyrazolines as
pharmacologically attractive scaffolds were described in a number of reviews in which the …
pharmacologically attractive scaffolds were described in a number of reviews in which the …
Thermal properties, antimicrobial activity and DNA binding of Ni (II) complexes of azo dye compounds
A novel series of nickel (II) azo dye complexes of 5-(4-methoxyphenylazo)-2-thioxo-4-
thiazolidinone (HL 1), 5-(4-methylphenylazo)-2-thioxo-4-thiazolidinone (HL 2), 5 …
thiazolidinone (HL 1), 5-(4-methylphenylazo)-2-thioxo-4-thiazolidinone (HL 2), 5 …
Synthesis, characterization, DNA binding and antitumor activities of Cu (II) complexes
A series of Cu (II) complexes of 5, 5-dimethyl-2-(2-arylhydrazono) cyclohexane-1, 3-dione
(HL n) were synthesized by the coupling of dimedone with aniline and its derivatives. These …
(HL n) were synthesized by the coupling of dimedone with aniline and its derivatives. These …
[PDF][PDF] Antibacterial activity of thiazole and its derivatives
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
Influence of substituent effects on spectroscopic properties and antimicrobial activity of 5-(4′-substituted phenylazo)-2-thioxothiazolidinone derivatives
Abstract 5-(4′-substituted phenylazo)-2-thioxothiazolidinone derivatives (HL n) have been
synthesized and characterized by elemental analysis, spectra (IR, electronic and 1 H NMR) …
synthesized and characterized by elemental analysis, spectra (IR, electronic and 1 H NMR) …
Synthesis and structure–activity-relationship studies of thiazolidinediones as antiplasmodial inhibitors of the Plasmodium falciparum cysteine protease falcipain-2
Following a structure-based virtual screening, a series of 2, 4 thiazolidinediones was
synthesized in order to explore structure activity relationships for inhibition of the …
synthesized in order to explore structure activity relationships for inhibition of the …
Synthesis, anticancer assessment on human breast, liver and colon carcinoma cell lines and molecular modeling study using novel pyrazolo [4, 3-c] pyridine …
NH Metwally, EA Deeb - Bioorganic Chemistry, 2018 - Elsevier
Abstract The key intermediate 3-aminopyrazolo [4, 3-c] pyridine-4, 6-dione (2) is considered
as a precursor for some novel pyrazolo [4, 3-c] pyridines 4a-c, arylhydrazopyrazolo [4, 3-c] …
as a precursor for some novel pyrazolo [4, 3-c] pyridines 4a-c, arylhydrazopyrazolo [4, 3-c] …
Synthesis, biological evaluation of novel thiopyrano [2, 3-d] thiazoles incorporating arylsulfonate moiety as potential inhibitors of tubulin polymerization, and molecular …
NH Metwally, MA Badawy, DS Okpy - Journal of Molecular Structure, 2022 - Elsevier
Abstract Novel series of thiopyrano [2, 3-d] 1, 3-thiazole derivatives incorporating
arylsulfonate moiety were synthesized and characterized by 1 H NMR, 13 C NMR, MS, and …
arylsulfonate moiety were synthesized and characterized by 1 H NMR, 13 C NMR, MS, and …