Quinazolinone and quinazoline derivatives: recent structures with potent antimicrobial and cytotoxic activities

E Jafari, MR Khajouei, F Hassanzadeh… - Research in …, 2016 - journals.lww.com
The heterocyclic compounds have a great importance in medicinal chemistry. One of the
most important heterocycles in medicinal chemistry are quinazolines possessing wide …

A review: Structure-activity relationship and antibacterial activities of Quinoline based hybrids

KB Patel, P Kumari - Journal of Molecular Structure, 2022 - Elsevier
The drug resistance problem is most acute in the case of bacteria. There is always a need to
develop novel antibacterial drugs with better mechanisms of action. Most of the quinoline …

Current perspectives on quinazolines with potent biological activities: A review

T Gupta, A Rohilla, A Pathak, MJ Akhtar… - Synthetic …, 2018 - Taylor & Francis
Quinazoline is a heterocyclic compound having biological activities. It is aromatic in nature
having bicyclic structure containing benzene ring and pyrimidine ring. Quinazoline and its …

Hybrid bioactive heterocycles as potential antimicrobial agents: a review

N Desai, A Trivedi, U Pandit, A Dodiya… - Mini Reviews in …, 2016 - ingentaconnect.com
The ever increasing cases of microbial resistance pose a major threat to the scientific
community and therefore the need for discovery and development of newer antimicrobial …

Design, synthesis, antimicrobial evaluation, and molecular docking study of some 4-thiazolidinone derivatives containing pyridine and quinazoline moiety

NC Desai, KA Jadeja, DJ Jadeja… - Synthetic …, 2021 - Taylor & Francis
Abstract A series of 5-aryl-3-(4-oxo-2-phenylquinazolin-3 (4 H)-yl)-2-(pyridin-4-yl) thiazolidin-
4-ones were synthesized and evaluated for their antibacterial and antifungal activities …

A visible light mediated, metal and oxidant free highly efficient cross dehydrogenative coupling (CDC) reaction between quinoxalin-2 (1 H)-ones and ethers

KD Mane, RB Kamble, G Suryavanshi - New Journal of Chemistry, 2019 - pubs.rsc.org
The efficient and metal free, white light mediated 3C alkylation of quinoxalin-2 (1H)-ones via
a cross dehydrogenative coupling reaction with cyclic ethers using eosin Y as a …

Synthesis, spectroscopic characterization, DFT, molecular docking and in vitro antibacterial potential of novel quinoline derivatives

Y Bouzian, Y Sert, K Khalid, L Van Meervelt… - Journal of Molecular …, 2021 - Elsevier
In this work, three new quinolone derivatives were prepared by alkylation of 2-oxo-1, 2-
dihydroquinoline-4-carboxylic acid with ethyl 2-bromoacetate. The synthesized compounds …

[PDF][PDF] Synthetic and therapeutic potential of 4-thiazolidinone and its analogs

N Agrawal - Curr Chem Lett, 2021 - pdfs.semanticscholar.org
The chemistry of five-membered rings containing two heteroatoms has been an interesting
field of study for decades. Among which 4-thiazolidinone ring system 1 has been studied …

Chemistry of quinolines and their agrochemical potential

D Utreja, R Salotra, G Kaur, S Sharma… - Current Organic …, 2022 - benthamdirect.com
Human population is increasing at an alarming rate which indirectly imposes pressure on
agriculture and food supply. However, crop production is reduced by pathogenic infections …

Importance of quinazoline and quinazolinone derivatives in medicinal chemistry

M Bhat, SL Belagali, SV Mamatha, BK Sagar… - Studies in Natural …, 2021 - Elsevier
The compounds of the quinazoline family belong to the nitrogen-containing heterocyclics;
the core structure represents various biological activities, and many natural compounds are …