Isocyanide-based multicomponent reactions for the synthesis of benzopyran derivatives with biological scaffolds

MT Nazeri, T Nasiriani, S Torabi… - Organic & Biomolecular …, 2024 - pubs.rsc.org
Benzopyrans (BZPs) are one of the most privileged and influential small O-heterocycles that
form the core of many natural compounds, commercial drugs, biological compositions …

Dual active 1, 4-dihydropyridine derivatives: Design, green synthesis and in vitro anti-cancer and anti-oxidant studies

P Anaikutti, P Makam - Bioorganic Chemistry, 2020 - Elsevier
The present work describes the design of 1, 4-dihydropyridines (1, 4-DHPs) with diverse
variations in structural and functional groups. The physico-chemical properties and drug-like …

Indolyl-4H-chromenes: Multicomponent one-pot green synthesis, in vitro and in silico, anticancer and antioxidant studies

P Anaikutti, M Selvaraj, J Prabhakaran… - Journal of Molecular …, 2022 - Elsevier
The present work describes the simple, economical and eco-friendly multicomponent one-
pot synthesis of indolyl-4H-chromene derivatives. It is being achieved by reacting …

[HTML][HTML] Antibacterial and antioxidant potential of GC-MS analysis of crude ethyl acetate extract from the tropical mangrove plant Avicennia officinalis L.

P Lalitha, A Parthiban, V Sachithanandam… - South African Journal of …, 2021 - Elsevier
Avicennia officinalis L. is an important mangrove plant used in traditional medicine to treat
various diseases like asthma, dyspepsia, paralysis, tumor and rheumatism in aboriginal …

Synthesis, in vitro, in silico and DFT studies of indole curcumin derivatives as potential anticancer agents

A Parthiban, R Sivasankar, B Rajdev, RN Asha… - Journal of Molecular …, 2022 - Elsevier
The curcumin derivatives were synthesized for the first time using simple starting materials
through a three-component reaction, yielding high purity compounds. The synthesized …

Iodine catalyzed synthesis of imidazo [1, 2-a] pyrazine and imidazo [1, 2-a] pyridine derivatives and their anticancer activity

R Krishnamoorthy, P Anaikutti - RSC advances, 2023 - pubs.rsc.org
An efficient iodine-catalyzed method for synthesizing imidazo [1, 2-a] pyrazines and imidazo
[1, 2-a] pyridines via one-pot three-component condensations has been reported. The …

Green synthesis of gold nanoparticles using quercetin biomolecule from mangrove plant, Ceriops tagal: Assessment of antiproliferative properties, cellular uptake and …

A Parthiban, V Sachithanandam… - Journal of Molecular …, 2023 - Elsevier
Synthesis, structural elucidation and in vitro cytotoxic properties of quercetin gold
nanoparticles (Qu-AuNPs) were derived from the mangrove plant, Ceriops tagal. UV–Visible …

A comprehensive in silico and in vitro studies on quinizarin: a promising phytochemical derived from Rhizophora mucronata Lam

V Sachithanandam, P Lalitha, A Parthiban… - Journal of …, 2022 - Taylor & Francis
Mangrove plants are a great source of phytomedicines, since from the beginning of human
civilization and the origin of traditional medicines. In the present study, ten different …

Anticancer activities, molecular docking and structure–activity relationship of novel synthesized 4H-chromene, and 5H-chromeno[2,3-d]pyrimidine candidates

AH Halawa, MM Elaasser, AM El Kerdawy… - Medicinal Chemistry …, 2017 - Springer
In the present study, a series of 4 H-chromene and 5 H-chromeno [2, 3-d] pyrimidine
derivatives was synthesized and evaluated as potential cytotoxic agents. The cytotoxic …

Synthesis, in vitro and in silico antimalarial activity of 7-chloroquinoline and 4H-chromene conjugates

A Parthiban, J Muthukumaran, A Manhas… - Bioorganic & medicinal …, 2015 - Elsevier
A new series of chloroquinoline-4H-chromene conjugates incorporating piperizine or
azipane tethers were synthesized and their anti-malarial activity were evaluated against two …