Prospective of 68Ga-radiopharmaceutical development

I Velikyan - Theranostics, 2013 - pmc.ncbi.nlm.nih.gov
Positron Emission Tomography (PET) experienced accelerated development and has
become an established method for medical research and clinical routine diagnostics on …

PET radiopharmaceuticals for imaging of tumor hypoxia: a review of the evidence

E Lopci, I Grassi, A Chiti, C Nanni… - American journal of …, 2014 - pmc.ncbi.nlm.nih.gov
Hypoxia is a pathological condition arising in living tissues when oxygen supply does not
adequately cover the cellular metabolic demand. Detection of this phenomenon in tumors is …

The ubiquitous DOTA and its derivatives: the impact of 1, 4, 7, 10-tetraazacyclododecane-1, 4, 7, 10-tetraacetic acid on biomedical imaging

GJ Stasiuk, NJ Long - Chemical Communications, 2013 - pubs.rsc.org
Over the last twenty-five years 1, 4, 7, 10-tetraazacyclododecane-1, 4, 7, 10-tetraacetic acid
(DOTA) has made a significant impact on the field of diagnostic imaging. DOTA is not the …

Advances in PET and MRI imaging of tumor hypoxia

P Gouel, P Decazes, P Vera, I Gardin, S Thureau… - Frontiers in …, 2023 - frontiersin.org
Tumor hypoxia is a complex and evolving phenomenon both in time and space. Molecular
imaging allows to approach these variations, but the tracers used have their own limitations …

Bifunctional gallium-68 chelators: Past, present, and future

P Spang, C Herrmann, F Roesch - Seminars in nuclear medicine, 2016 - Elsevier
This article reviews the development of bifunctional chelates for synthesising 68 Ga
radiopharmaceuticals. It structures the chelates into groups of macrocycles …

Metal-based redox-responsive MRI contrast agents

SM Pinto, V Tomé, MJF Calvete, MMCA Castro… - Coordination Chemistry …, 2019 - Elsevier
Given their potential in a better characterization and diagnosis of major pathologies like
cancer or chronic inflammation, redox-activated Magnetic Resonance Imaging (MRI) probes …

Longitudinal PET imaging of tumor hypoxia during the course of radiotherapy

S Stieb, A Eleftheriou, G Warnock… - European journal of …, 2018 - Springer
Hypoxia results from an imbalance between oxygen supply and consumption. It is a
common phenomenon in solid malignant tumors such as head and neck cancer. As hypoxic …

Redox‐and hypoxia‐responsive MRI contrast agents

QN Do, JS Ratnakar, Z Kovács, AD Sherry - ChemMedChem, 2014 - Wiley Online Library
The development of responsive or “smart” magnetic resonance imaging (MRI) contrast
agents that can report specific biomarker or biological events has been the focus of MRI …

Scandium-44: diagnostic feasibility in tumor-related angiogenesis

G Trencsényi, Z Képes - International Journal of Molecular Sciences, 2023 - mdpi.com
Angiogenesis-related cell-surface molecules, including integrins, aminopeptidase N,
vascular endothelial growth factor, and gastrin-releasing peptide receptor (GRPR), play a …

Molecular imaging of tumor hypoxia: Evolution of nitroimidazole radiopharmaceuticals and insights for future development

S Mittal, MB Mallia - Bioorganic Chemistry, 2023 - Elsevier
Though growing evidence has been collected in support of the concept of dose escalation
based on the molecular level images indicating hypoxic tumor sub-volumes that could be …