Advances in the structure, mechanism and targeting of chemoresistance-linked ABC transporters

A Sajid, H Rahman, SV Ambudkar - Nature Reviews Cancer, 2023‏ - nature.com
Cancer cells frequently display intrinsic or acquired resistance to chemically diverse
anticancer drugs, limiting therapeutic success. Among the main mechanisms of this …

Chemical molecular‐based approach to overcome multidrug resistance in cancer by targeting P‐glycoprotein (P‐gp)

H Zhang, H Xu, CR Ashby Jr, YG Assaraf… - Medicinal research …, 2021‏ - Wiley Online Library
Multidrug resistance (MDR) remains one of the major impediments for efficacious cancer
chemotherapy. Increased efflux of multiple chemotherapeutic drugs by transmembrane ATP …

Multidrug resistance proteins (MRPs): Structure, function and the overcoming of cancer multidrug resistance

JQ Wang, Y Yang, CY Cai, QX Teng, Q Cui, J Lin… - Drug Resistance …, 2021‏ - Elsevier
ATP-binding cassette (ABC) transporters mediate the ATP-driven translocation of structurally
and mechanistically distinct substrates against steep concentration gradients. Among the …

ATP‐binding cassette (ABC) transporters in cancer: A review of recent updates

JQ Wang, ZX Wu, Y Yang, QX Teng… - Journal of Evidence …, 2021‏ - Wiley Online Library
The ATP‐binding cassette (ABC) transporter superfamily is one of the largest membrane
protein families existing in wide spectrum of organisms from prokaryotes to human. ABC …

Structural and functional aspects of P-glycoprotein and its inhibitors

S Mollazadeh, A Sahebkar, F Hadizadeh, J Behravan… - Life sciences, 2018‏ - Elsevier
Abstract P-glycoprotein (P-gp) is a member of ATP-binding cassette (ABC) superfamily
which extrudes chemotherapeutic agents out of the cell. Suppression of this efflux activity …

Antibody-Free Fluorine-Assisted Metabolic Sequencing of RNA N4-Acetylcytidine

S Yan, Z Lu, W Yang, J Xu, Y Wang… - Journal of the …, 2023‏ - ACS Publications
N 4-Acetylcytidine (ac4C) has been found to affect a variety of cellular and biological
processes. For a mechanistic understanding of the roles of ac4C in biology and disease, we …

The role of ABCC10/MRP7 in anti-cancer drug resistance and beyond

DQ Chen, Y **e, LQ Cao, JS Fleishman, Y Chen… - Drug Resistance …, 2024‏ - Elsevier
Abstract Multidrug resistance protein 7 (MRP7), also known as ATP-binding cassette (ABC)
transporter subfamily C10 (ABCC10), is an ABC transporter that was first identified in 2001 …

Discovery of new 4-indolyl quinazoline derivatives as highly potent and orally bioavailable P-glycoprotein inhibitors

S Yuan, B Wang, QQ Dai, XN Zhang… - Journal of Medicinal …, 2021‏ - ACS Publications
The major drawbacks of P-glycoprotein (P-gp) inhibitors at the clinical stage make the
development of new P-gp inhibitors challenging and desirable. In this study, we reported our …

Evaluation of the FDA-approved kinase inhibitors to uncover the potential repurposing candidates targeting ABC transporters in multidrug-resistant cancer cells: an in …

A Poustforoosh, F Moosavi - Journal of Biomolecular Structure and …, 2024‏ - Taylor & Francis
Multiple drug resistance (MDR) is characterized by the resistance of cancer cells to a broad
spectrum of anticancer drugs. The main mechanism underlying the MDR phenotype is the …

Lysine-specific demethylase 1 promises to be a novel target in cancer drug resistance: therapeutic implications

FF Yang, XL Xu, T Hu, JQ Liu, JZ Zhou… - Journal of Medicinal …, 2023‏ - ACS Publications
Chemotherapy, targeted therapy, and immunotherapy are effective against most tumors, but
drug resistance remains a barrier to successful treatment. Lysine-specific demethylase 1 …