Chromone: a valid scaffold in medicinal chemistry

A Gaspar, MJ Matos, J Garrido, E Uriarte… - Chemical …, 2014 - ACS Publications
Chromones are a group of naturally occurring compounds that are ubiquitous in nature,
especially in plants. The word chromone is derived from the Greek word chroma, meaning …

Chromones as a privileged scaffold in drug discovery: A review

RS Keri, S Budagumpi, RK Pai… - European Journal of …, 2014 - Elsevier
The chromone and its derivatives are the most important heterocyclic compounds, which is a
common and integral feature of a variety of natural products and medicinal agents. These …

Cytotoxic activity of 3-(5-phenyl-3H-[1, 2, 4] dithiazol-3-yl) chromen-4-ones and 4-oxo-4H-chromene-3-carbothioic acid N-phenylamides

T Raj, RK Bhatia, M Sharma, AK Saxena… - European journal of …, 2010 - Elsevier
6/6, 7-Substituted-3-formylchromones (8a–g) were reacted with 2 equivalents
thiobenzamide (9) in refluxing toluene to furnish substituted-3-(5-phenyl-3H-[1, 2, 4] dithiazol …

An update on natural occurrence and biological activity of chromones

SK Sharma, S Kumar, K Chand… - Current medicinal …, 2011 - ingentaconnect.com
The chemistry of chromones is very well known. This system is widely used in organic
chemistry as an intermediate compound for the synthesis of numerous hetrocycles. On the …

One-pot synthesis of dihydropyrano [2, 3-c] chromenes via a three component coupling of aromatic aldehydes, malononitrile, and 3-hydroxycoumarin catalyzed by …

S Paul, P Bhattacharyya, AR Das - Tetrahedron Letters, 2011 - Elsevier
An efficient and green protocol for the synthesis of dihydropyrano [2, 3-c] chromene
derivatives by one-pot, three component coupling reaction of aromatic aldehyde …

Synthesis, structure–activity relationship of novel substituted 4H-chromen-1, 2, 3, 4-tetrahydropyrimidine-5-carboxylates as potential anti-mycobacterial and anticancer …

BC Raju, RN Rao, P Suman, P Yogeeswari… - Bioorganic & Medicinal …, 2011 - Elsevier
Abstract Series of 4H-chromen-1, 2, 3, 4-tetrahydropyrimidine-5-carboxylate derivatives 7a–
7zb, 8a–8d and 9a–9d were synthesized and screened for their in vitro anti-mycobacterial …

Design, Synthesis, Biological Evaluation, and Molecular Modeling of Novel 4H-Chromene Analogs as Potential Succinate Dehydrogenase Inhibitors

T Lu, Y Yan, T Zhang, G Zhang, T **ao… - Journal of Agricultural …, 2021 - ACS Publications
Thirty-one new 4 H-chromene derivatives were designed and synthesized. Their structures
were identified with IR, 1H NMR, 13C NMR, and HRMS. The crystal structure of compound …

Recyclizations of 3-formylchromones with binucleophiles

AS Plaskon, OO Grygorenko, SV Ryabukhin - Tetrahedron, 2012 - Elsevier
Chromones are widely recognized as an important class of biologically active compounds of
both natural and synthetic origin. 1 e8 The less known but very useful application of the …

Highly efficient three-component, one-pot synthesis of dihydropyrano[3,2-c]chromene derivatives

HJ Wang, J Lu, ZH Zhang - Monatshefte für Chemie-Chemical Monthly, 2010 - Springer
An efficient and convenient method for synthesis of dihydropyrano [3, 2-c] chromene
derivatives by one-pot, three-component reaction of aldehydes, malononitrile, and 4 …

Magnetically retrievable nano crystalline CuFe 2 O 4 catalyzed multi-component reaction: a facile and efficient synthesis of functionalized dihydropyrano [2, 3-c] …

K Pradhan, S Paul, AR Das - Catalysis Science & Technology, 2014 - pubs.rsc.org
CuFe2O4 magnetic nanoparticles were synthesized and recognized as an efficient catalyst
for the one-pot synthesis of dihydropyrano [2, 3-c] pyrazole, pyrano [3, 2-c] coumarin and 4H …