[HTML][HTML] Implications of NQO1 in cancer therapy

ET Oh, HJ Park - BMB reports, 2015‏ - ncbi.nlm.nih.gov
Abstract NAD (P) H: quinone oxidoreductase (NQO1), an obligatory two-electron reductase,
is a ubiquitous cytosolic enzyme that catalyzes the reduction of quinone substrates. The …

The protective effect of natural compounds against rotenone‐induced neurotoxicity

F Yarmohammadi, A Wallace Hayes… - … of Biochemical and …, 2020‏ - Wiley Online Library
Rotenone is a widely used organic pesticide; its serious side effect for off‐target species is
neurotoxicity. The primary mechanism of rotenone toxicity is inhibition of the mitochondrial …

Lipophilicity, pharmacokinetic properties, and molecular docking study on SARS-CoV-2 target for betulin triazole derivatives with attached 1, 4-quinone

M Kadela-Tomanek, M Jastrzębska, K Marciniec… - Pharmaceutics, 2021‏ - mdpi.com
A key parameter in the design of new active compounds is lipophilicity, which influences the
solubility and permeability through membranes. Lipophilicity affects the pharmacodynamic …

The potential of Ginkgo biloba in the treatment of human diseases and the relationship to Nrf2–mediated antioxidant protection

Y Li, X Zhu, K Wang, L Zhu, M Murray… - Journal of Pharmacy …, 2022‏ - academic.oup.com
Objectives This review summarises the current findings regarding the therapeutic effects of
GBE and its active ingredients in relation to the Nrf2 antioxidant cascade, to provide …

The effects of in ovo feeding of selenized glucose on selenium concentration and antioxidant capacity of breast muscle in neonatal broilers

M Zhao, J Li, Q Shi, H Shan, L Liu, T Geng, L Yu… - … Trace Element Research, 2023‏ - Springer
This study aims to investigate the impacts of in ovo feeding (IOF) of selenized glucose
(SeGlu) on selenium (Se) level and antioxidant capacity of breast muscle in newborn …

Association of Genetic Variations in NRF2, NQO1, HMOX1, and MT with Severity of Coronary Artery Disease and Related Risk Factors

I Sarutipaiboon, N Settasatian, N Komanasin… - Cardiovascular …, 2020‏ - Springer
NRF2 is a transcription factor which, during oxidative stress, activates transcription of its
target antioxidant genes. Polymorphisms in NRF2 and its target antioxidant genes: HMOX-1 …

Флавоноиды глазами фармаколога. Антиоксидантная и противовоспалительная активность

ЯФ Зверев - Обзоры по клинической фармакологии и …, 2017‏ - cyberleninka.ru
Обзор литературы посвящен рассмотрению механизмов антиоксидантного и
противовоспалительного действия флавоноидов. При обсуждении антиоксидантного …

6-Shogaol inhibits advanced glycation end-products-induced IL-6 and ICAM-1 expression by regulating oxidative responses in human gingival fibroblasts

K Nonaka, M Bando, E Sakamoto, Y Inagaki… - Molecules, 2019‏ - mdpi.com
Advanced glycation end-products (AGEs) cause diabetes mellitus (DM) complications and
accumulate more highly in periodontal tissues of patients with periodontitis and DM. AGEs …

Design, synthesis and biological activity of 1, 4-quinone moiety attached to betulin derivatives as potent DT-diaphorase substrate

M Kadela-Tomanek, M Jastrzębska, K Marciniec… - Bioorganic …, 2021‏ - Elsevier
In this research, betulin derivatives were bonded to the 1, 4-quinone fragment by triazole
linker. Furthermore, the enzymatic assay used has shown that these compounds are a good …

The GTPase KRAS suppresses the p53 tumor suppressor by activating the NRF2-regulated antioxidant defense system in cancer cells

H Yang, S **ang, A Kazi, SM Sebti - Journal of Biological Chemistry, 2020‏ - ASBMB
In human cancer cells that harbor mutant KRAS and WT p53 (p53), KRAS contributes to the
maintenance of low p53 levels. Moreover, KRAS depletion stabilizes and reactivates p53 …