Asymmetric one-pot synthesis of 1, 3-oxazolidines and 1, 3-oxazinanes via hemiaminal intermediates

SK Nimmagadda, Z Zhang, JC Antilla - Organic Letters, 2014‏ - ACS Publications
A highly efficient method for the enantioselective one-pot synthesis of 1, 3-oxazolidines and
1, 3-oxazinanes has been reported. The reaction proceeds via the formation of hemiaminal …

New Zealand glowworm (Arachnocampa luminosa) bioluminescence is produced by a firefly-like luciferase but an entirely new luciferin

OC Watkins, ML Sharpe, NB Perry, KL Krause - Scientific Reports, 2018‏ - nature.com
Abstract The New Zealand glowworm, Arachnocampa luminosa, is well-known for displays
of blue-green bioluminescence, but details of its bioluminescent chemistry have been …

Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity

M Meldal, CW Tornøe, TE Nielsen… - Peptide Science …, 2010‏ - Wiley Online Library
A huge unleashed potential lies hidden in the large and diverse pool of encoded and
particularly nonencoded chiral α‐, β‐, and γ‐amino acids available today. Although these …

Efficient Solid‐Phase Synthesis of Peptide‐Based Phosphine Ligands: Towards Combinatorial Libraries of Selective Transition Metal Catalysts

CA Christensen, M Meldal - Chemistry–A European Journal, 2005‏ - Wiley Online Library
A new methodology for the solid‐phase synthesis of peptide‐based phosphine ligands has
been developed. Solid supported peptide scaffolds possessing either primary or secondary …

Solid‐Phase Synthesis of Tetrahydro‐β‐carbolines and Tetrahydroisoquinolines by Stereoselective Intramolecular N‐Carbamyliminium Pictet–Spengler Reactions

F Diness, J Beyer, M Meldal - Chemistry–A European Journal, 2006‏ - Wiley Online Library
A solid‐phase method for the synthesis of tri‐, tetra‐, and pentacyclic compounds containing
tetrahydro‐β‐carboline, tetrahydroisoquinoline or analogous scaffolds is presented. The …

Facile synthesis of SAM–peptide conjugates through alkyl linkers targeting protein N-terminal methyltransferase 1

G Zhang, R Huang - RSC advances, 2016‏ - pubs.rsc.org
We report the first chemical synthesis of SAM–peptide conjugates through alkyl linkers to
prepare bisubstrate analogs for protein methyltransferases. We demonstrate its application …

Solid-phase synthesis of a peptide-based P, S-ligand system designed for generation of combinatorial catalyst libraries

CA Christensen, M Meldal - Journal of Combinatorial Chemistry, 2007‏ - ACS Publications
An efficient methodology for the solid-phase synthesis of diverse combinatorial peptide-
based P, S-ligand libraries based on a modular approach was developed. Chiral thioethers …

Versatile Synthesis of Free and N‐Benzyloxycarbonyl‐Protected 2,2‐Disubstituted Taurines

B Wang, W Zhang, L Zhang, DM Du, G Liu, J Xu - 2008‏ - Wiley Online Library
An effective and versatile method was developed to synthesize N‐benzyloxycarbonyl‐
protected and free 2, 2‐disubstituted taurines. Several novel 2, 2‐disubstituted taurines …

Diversity‐Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides

Y Wang, AØ Madsen, F Diness… - Chemistry–A European …, 2017‏ - Wiley Online Library
Cascade reactions proceeding through peptide‐derived N‐carbamoyl iminium ions are
reported. Two new reactions of N‐carbamoyl iminium ions are described, including a …

Efficient 'one-pot'methodology for the synthesis of novel tetrahydro-β-carboline, tetrahydroisoquinoline and tetrahydrothienopyridine derivatives

A Ionescu, D Cornut, S Soriano, C Guissart… - Tetrahedron …, 2013‏ - Elsevier
A simple and efficient 'one-pot'methodology was developed to generate a new series of
tetrahydro-β-carboline (THBC), tetrahydroisoquinoline (THIQ) and tetrahydrothienopyridine …