Computer aided drug design for multi-target drug design: SAR/QSAR, molecular docking and pharmacophore methods

A Abdolmaleki, JB Ghasemi… - Current Drug Targets, 2017‏ - ingentaconnect.com
Multi-target drugs against particular multiple targets get better protection, resistance profiles
and curative influence by cooperative rules of a key beneficial target with resistance …

Multivariate statistical analysis methods in QSAR

S Pirhadi, F Shiri, JB Ghasemi - Rsc Advances, 2015‏ - pubs.rsc.org
The emphasis of this review is particularly on multivariate statistical methods currently used
in quantitative structure–activity relationship (QSAR) studies. The mathematical methods for …

Innovative screening for functional improved aromatic amine derivatives: Toxicokinetics, free radical oxidation pathway and carcinogenic adverse outcome pathway

Y Liu, X Li, Q Pu, R Fu, Z Wang, Y Li, X Li - Journal of Hazardous Materials, 2023‏ - Elsevier
Aromatic amines, one of the most widely used low-cost antioxidants in rubbers, have been
regarded as pollutants with human health concerns. To overcome this problem, this study …

Computational approaches for the design of novel dopamine D2 and serotonin 5-HT2A receptor dual antagonist towards schizophrenia

A Rathore, V Asati, M Mishra, R Das, V Kashaw… - In Silico …, 2022‏ - Springer
Piperidine and piperazine derivatives exhibit a diverse range of biological applications,
including antipsychotic activity. In this study, a dataset of molecules containing piperidine …

Methods and applications of structure based pharmacophores in drug discovery

S Pirhadi, F Shiri, JB Ghasemi - Current topics in medicinal …, 2013‏ - ingentaconnect.com
A pharmacophore model does not describe a real molecule or a real association of
functional groups but illustrates a molecular recognition of a biological target shared by a …

Computer-aided drug discovery approaches against the tropical infectious diseases malaria, tuberculosis, trypanosomiasis, and leishmaniasis

PM Njogu, EM Guantai, E Pavadai… - ACS infectious …, 2016‏ - ACS Publications
Despite the tremendous improvement in overall global health heralded by the adoption of
the Millennium Declaration in the year 2000, tropical infections remain a major health …

The advancement of multidimensional QSAR for novel drug discovery-where are we headed?

T Wang, X Yuan, MB Wu, JP Lin… - Expert opinion on drug …, 2017‏ - Taylor & Francis
ABSTRACT Introduction: The Multidimensional quantitative structure− activity relationship
(multidimensional-QSAR) method is one of the most popular computational methods …

Dual-acting of hybrid compounds-a new dawn in the discovery of multi-target drugs: lead generation approaches

A Abdolmaleki, JB Ghasemi - Current Topics in Medicinal …, 2017‏ - ingentaconnect.com
Finding high quality beginning compounds is a critical job at the start of the lead generation
stage for multi-target drug discovery (MTDD). Designing hybrid compounds as selective …

Targeting cysteine proteases from Plasmodium falciparum: A general overview, rational drug design and computational approaches for drug discovery

BD Bekono, F Ntie-Kang, LC Owono Owono… - Current Drug …, 2018‏ - benthamdirect.com
Background: The Plasmodium falciparum cysteine proteases, also known as falcipains, are
involved in different erythrocytic cycle processes of the malaria parasite, eg hydrolysis of …

Understanding chemico‐biological interactions of glutamate MMP‐2 inhibitors through rigorous alignment‐dependent 3D‐QSAR analyses

N Adhikari, SA Amin, A Saha, T Jha - ChemistrySelect, 2017‏ - Wiley Online Library
The current study involves different alignment techniques (pharmacophore‐based, docking‐
based and Open3DALIGN‐based) extensively at the first time to build three‐dimensional …