PPARγ signaling and metabolism: the good, the bad and the future

M Ahmadian, JM Suh, N Hah, C Liddle, AR Atkins… - Nature medicine, 2013 - nature.com
Thiazolidinediones (TZDs) are potent insulin sensitizers that act through the nuclear
receptor peroxisome proliferator-activated receptor-γ (PPARγ) and are highly effective oral …

[HTML][HTML] PPARgamma in metabolism, immunity, and cancer: unified and diverse mechanisms of action

M Hernandez-Quiles, MF Broekema… - Frontiers in …, 2021 - frontiersin.org
The proliferator-activated receptor γ (PPARγ), a member of the nuclear receptor superfamily,
is one of the most extensively studied ligand-inducible transcription factors. Since its …

The selection and function of cell type-specific enhancers

S Heinz, CE Romanoski, C Benner… - Nature reviews Molecular …, 2015 - nature.com
The human body contains several hundred cell types, all of which share the same genome.
In metazoans, much of the regulatory code that drives cell type-specific gene expression is …

Transcriptional control of energy metabolism by nuclear receptors

C Scholtes, V Giguère - Nature reviews Molecular cell biology, 2022 - nature.com
Transcriptional regulation of catabolic pathways is a central mechanism by which cells
respond to physiological cues to generate the energy required for anabolic pathways …

[HTML][HTML] Remodeling of the enhancer landscape during macrophage activation is coupled to enhancer transcription

MU Kaikkonen, NJ Spann, S Heinz, CE Romanoski… - Molecular cell, 2013 - cell.com
Recent studies suggest a hierarchical model in which lineage-determining factors act in a
collaborative manner to select and prime cell-specific enhancers, thereby enabling signal …

PPARγ and the global map of adipogenesis and beyond

MI Lefterova, AK Haakonsson, MA Lazar… - Trends in Endocrinology …, 2014 - cell.com
Peroxisome proliferator-activated receptor γ (PPARγ) is a member of the nuclear receptor
(NR) superfamily of ligand-dependent transcription factors (TFs) and function as a master …

Distinct but complementary contributions of PPAR isotypes to energy homeostasis

V Dubois, J Eeckhoute, P Lefebvre… - The Journal of clinical …, 2017 - Am Soc Clin Investig
Peroxisome proliferator–activated receptors (PPARs) regulate energy metabolism and
hence are therapeutic targets in metabolic diseases such as type 2 diabetes and non …

PPARs: fatty acid sensors controlling metabolism

L la Cour Poulsen, M Siersbæk, S Mandrup - Seminars in cell & …, 2012 - Elsevier
The peroxisome proliferator activated receptors (PPARs) are nuclear receptors that play key
roles in the regulation of lipid metabolism, inflammation, cellular growth, and differentiation …

Transcriptional and epigenetic control of brown and beige adipose cell fate and function

T Inagaki, J Sakai, S Kajimura - Nature reviews Molecular cell biology, 2016 - nature.com
White adipocytes store excess energy in the form of triglycerides, whereas brown and beige
adipocytes dissipate energy in the form of heat. This thermogenic function relies on the …

PPAR agonists and metabolic syndrome: an established role?

M Botta, M Audano, A Sahebkar, CR Sirtori… - International journal of …, 2018 - mdpi.com
Therapeutic approaches to metabolic syndrome (MetS) are numerous and may target
lipoproteins, blood pressure or anthropometric indices. Peroxisome proliferator-activated …