A review on the chemistry, coordination, structure and biological properties of 1-(acyl/aroyl)-3-(substituted) thioureas

A Saeed, U Flörke, MF Erben - Journal of Sulfur Chemistry, 2014 - Taylor & Francis
This review provides an overview of the chemistry, structure and potential applications of 1-
(acyl/aroyl)-3-(mono-substituted) and 1-(acyl/aroyl)-3, 3-(di-substituted) thioureas, with …

Recent advances in urea-and thiourea-based metal complexes: biological, sensor, optical, and corroson inhibition studies

RK Mohapatra, PK Das, MK Pradhan… - Comments on …, 2019 - Taylor & Francis
Ureas and thioureas, otherwise known as carbamides and thiocarbamides, respectively, are
rich sources of nitrogen. Urea has a wide range of applications in agriculture, the chemical …

Design, synthesis, characterization, and biological evaluation of nicotinoyl thioureas as antimicrobial and antioxidant agents

B Özgeriş - The Journal of Antibiotics, 2021 - nature.com
Addressed herein a series of thioureas starting from various amines and nicotinic acid have
been synthesized. Notably, thiourea based scaffolds are increasingly employed in medicinal …

Synthesis and bacteriostatic activities of bis (thiourea) derivatives with variable chain length

AN Abd Halim, Z Ngaini - Journal of Chemistry, 2016 - Wiley Online Library
A series of 1, 4‐bis (decoxyphenyl) carbamothioyl‐terephthalamide derivatives was
successfully synthesised by reaction of benzene‐1, 4‐dicarbonyl isothiocyanate …

Spectral characterization, DFT, docking and cytotoxicity of N-benzyl-4, 5-dihydro-3-methyl-5-oxo-1H-pyrazole-4-carbothioamide and its metal complexes

NM Hosny, A Belal, R Motawea, MA Hussien… - Journal of Molecular …, 2021 - Elsevier
A new ligand N-benzyl-4, 5-dihydro-3-methyl-5-oxo-1H-pyrazole-4-carbothioamide (H 2 L)
and some of its divalent metal complexes were synthesized. Elemental analyses, mass …

[PDF][PDF] Synthesis, crystal structure and in vitro anti-proliferative activity of 2-[(4-acetylphenyl) carbamoyl] phenyl acetate

RA Mohamed-Ezzat, BM Kariuki… - Acta Crystallographica …, 2023 - journals.iucr.org
2-[(4-Acetylphenyl) carbamoyl] phenyl acetate, C17H15NO4, has been synthesized and
structurally characterized. In the structure, N—H⋯ O hydrogen-bonding interactions form …

Synthesis of substituted phenethylamine-based thioureas and their antimicrobial and antioxidant properties

B Özgeriş - Russian Journal of Organic Chemistry, 2021 - Springer
Thiourea-based scaffolds are increasingly used in medicinal chemistry owing to their
tunable structural properties. This study demonstrates the first examples of phenethylamine …

Novel synthetic monothiourea aspirin derivatives bearing alkylated amines as potential antimicrobial agents

NA Nordin, TW Chai, BL Tan, CL Choi… - Journal of …, 2017 - Wiley Online Library
A new series of aspirin bearing alkylated amines moieties 1–12 were synthesised by
reacting isothiocyanate with a series of aniline derivatives in overall yield of 16–56%. The …

Synthesis and characterization of halogenated bis (acylthiourea) derivatives and their antibacterial activities

AN Abd Halim, Z Ngaini - Phosphorus, Sulfur, and Silicon and the …, 2017 - Taylor & Francis
ABSTRACT A total of 12 bis (acylthiourea) derivatives with different pharmacophores have
been synthesized via nucleophilic substitution reaction of benzene-1, 4-dicarbonyl …

Synthesis and Anticancer Activities of 4‐[(Halophenyl) diazenyl] phenol and 4‐[(Halophenyl) diazenyl] phenyl Aspirinate Derivatives against Nasopharyngeal Cancer …

BK Ho, Z Ngaini, P Matthew Neilsen… - Journal of …, 2017 - Wiley Online Library
Aspirin and azo derivatives have been widely studied and have drawn considerable
attention due to diverse biological activities. In this study, a series of 4‐[(halophenyl) …