Bis-and trisindolylmethanes (BIMs and TIMs)

M Shiri, MA Zolfigol, HG Kruger… - Chemical …, 2010‏ - ACS Publications
The indole ring system is present in many natural products, pharmaceuticals,
agrochemicals, and other compounds of importance. 1–8 The indole unit forms the basis for …

Unlocking diversity: from simple to cutting-edge synthetic methodologies of bis (indolyl) methanes

P Teli, S Soni, S Teli, S Agarwal - Topics in Current Chemistry, 2024‏ - Springer
From a synthetic perspective, bis (indolyl) methanes have undergone extensive
investigation over the past two to three decades owing to their remarkable pharmacological …

Formulation, characterization and pulmonary deposition of nebulized celecoxib encapsulated nanostructured lipid carriers

RR Patlolla, M Chougule, AR Patel, T Jackson… - Journal of Controlled …, 2010‏ - Elsevier
The aim of the current study was to encapsulate celecoxib (Cxb) in the nanostructured lipid
carrier (Cxb-NLC) nanoparticles and evaluate the lung disposition of nanoparticles following …

Potentiating photodynamic therapy of ICG-loaded nanoparticles by depleting GSH with PEITC

H Hu, J Chen, H Yang, X Huang, H Wu, Y Wu, F Li, Y Yi… - Nanoscale, 2019‏ - pubs.rsc.org
Photodynamic therapy (PDT) is a clinically approved cancer treatment which utilizes reactive
oxygen species (ROS) to eradicate cancer cells. But the high concentration of GSH inside …

Old wine in new bottles: Drug repurposing in oncology

M Antoszczak, A Markowska, J Markowska… - European Journal of …, 2020‏ - Elsevier
Increasing costs, much time consumption and high risk of failure associated with the process
of de novo development of new anticancer drugs have prompted the pharmaceutical …

[HTML][HTML] Antitumor effect of thymoquinone combined with resveratrol on mice transplanted with breast cancer

OH Alobaedi, WH Talib, IA Basheti - Asian Pacific journal of tropical …, 2017‏ - Elsevier
Objective To test the anticancer potential activity of the combination of thymoquinone (TQ)
and resveratrol (RES) against breast cancer in mice. Methods The antiproliferative activity of …

Attenuation of multi-targeted proliferation-linked signaling by 3, 3′-diindolylmethane (DIM): from bench to clinic

S Banerjee, D Kong, Z Wang, B Bao, GG Hillman… - … Research/Reviews in …, 2011‏ - Elsevier
Emerging evidence provide credible support in favor of the potential role of bioactive
products derived from ingesting cruciferous vegetables such as broccoli, brussel sprouts …

[HTML][HTML] The mycelium of the Trametes versicolor synn. Coriolus versicolor (Turkey tail mushroom) exhibit anti-melanoma activity in vitro

R Lowenthal, M Taylor, JA Gidden, B Heflin… - Biomedicine & …, 2023‏ - Elsevier
Melanoma is one of the most aggressive forms of skin cancer and is characterized by high
metastatic potential. Despite improvements in early diagnosis and treatment, the mortality …

Organocatalytic enantioselective SN 1-type dehydrative nucleophilic substitution: access to bis (indolyl) methanes bearing quaternary carbon stereocenters

WR Zhu, Q Su, XY Deng, JS Liu, T Zhong, SS Meng… - Chemical …, 2022‏ - pubs.rsc.org
A highly general and straightforward approach to access chiral bis (indolyl) methanes (BIMs)
bearing quaternary stereocenters has been realized via enantioconvergent dehydrative …

Anticancer properties of indole compounds: mechanism of apoptosis induction and role in chemotherapy

A Ahmad, WA Sakr… - Current drug targets, 2010‏ - ingentaconnect.com
Indole compounds, obtained from cruciferous vegetables, have been investigated for their
putative anti-cancer properties. Studies with indole-3-carbinol (I3C) and its dimeric product …