Structure, function, and pharmacology of glutamate receptor ion channels

KB Hansen, LP Wollmuth, D Bowie, H Furukawa… - Pharmacological …, 2021‏ - Elsevier
Many physiologic effects of l-glutamate, the major excitatory neurotransmitter in the
mammalian central nervous system, are mediated via signaling by ionotropic glutamate …

Autoantibodies to synaptic receptors and neuronal cell surface proteins in autoimmune diseases of the central nervous system

J Dalmau, C Geis, F Graus - Physiological reviews, 2017‏ - journals.physiology.org
Investigations in the last 10 years have revealed a new category of neurological diseases
mediated by antibodies against cell surface and synaptic proteins. There are currently 16 …

Structure, function, and allosteric modulation of NMDA receptors

KB Hansen, F Yi, RE Perszyk, H Furukawa… - Journal of General …, 2018‏ - rupress.org
NMDA-type glutamate receptors are ligand-gated ion channels that mediate a Ca2+-
permeable component of excitatory neurotransmission in the central nervous system (CNS) …

The important role of zinc in neurological diseases

Z Li, Y Liu, R Wei, VW Yong, M Xue - Biomolecules, 2022‏ - mdpi.com
Zinc is one of the most abundant metal ions in the central nervous system (CNS), where it
plays a crucial role in both physiological and pathological brain functions. Zinc promotes …

Crystal structure of a heterotetrameric NMDA receptor ion channel

E Karakas, H Furukawa - Science, 2014‏ - science.org
N-Methyl-d-aspartate (NMDA) receptors belong to the family of ionotropic glutamate
receptors, which mediate most excitatory synaptic transmission in mammalian brains …

Glutamate receptor ion channels: structure, regulation, and function

SF Traynelis, LP Wollmuth, CJ McBain, FS Menniti… - Pharmacological …, 2010‏ - Elsevier
The mammalian ionotropic glutamate receptor family encodes 18 gene products that
coassemble to form ligand-gated ion channels containing an agonist recognition site, a …

NMDA receptor structures reveal subunit arrangement and pore architecture

CH Lee, W Lü, JC Michel, A Goehring, J Du, X Song… - Nature, 2014‏ - nature.com
Abstract N-methyl-d-aspartate (NMDA) receptors are Hebbian-like coincidence detectors,
requiring binding of glycine and glutamate in combination with the relief of voltage …

Molecular mechanism of ligand gating and opening of NMDA receptor

TH Chou, M Epstein, RG Fritzemeier, NS Akins… - Nature, 2024‏ - nature.com
Glutamate transmission and activation of ionotropic glutamate receptors are the fundamental
means by which neurons control their excitability and neuroplasticity. The N-methyl-d …

Molecular basis of NMDA receptor functional diversity

P Paoletti - European Journal of Neuroscience, 2011‏ - Wiley Online Library
NMDA receptors (NMDARs) form glutamate‐gated ion channels widely expressed in the
central nervous system and highly permeable to calcium ions. NMDARs have always …

Distinct functional and pharmacological properties of Triheteromeric GluN1/GluN2A/GluN2B NMDA receptors

KB Hansen, KK Ogden, H Yuan, SF Traynelis - Neuron, 2014‏ - cell.com
NMDA receptors are tetrameric ligand-gated ion channels comprised of GluN1, GluN2, and
GluN3 subunits. Two different GluN2 subunits have been identified in most NMDA receptor …