In silico methods and tools for drug discovery

B Shaker, S Ahmad, J Lee, C Jung, D Na - Computers in biology and …, 2021 - Elsevier
In the past, conventional drug discovery strategies have been successfully employed to
develop new drugs, but the process from lead identification to clinical trials takes more than …

An updated review of computer‐aided drug design and its application to COVID‐19

AB Gurung, MA Ali, J Lee, MA Farah… - BioMed research …, 2021 - Wiley Online Library
The recent outbreak of the deadly coronavirus disease 19 (COVID‐19) pandemic poses
serious health concerns around the world. The lack of approved drugs or vaccines continues …

Structure-based drug design with equivariant diffusion models

A Schneuing, C Harris, Y Du, K Didi… - Nature Computational …, 2024 - nature.com
Abstract Structure-based drug design (SBDD) aims to design small-molecule ligands that
bind with high affinity and specificity to pre-determined protein targets. Generative SBDD …

[HTML][HTML] A structure-based drug discovery paradigm

M Batool, B Ahmad, S Choi - International journal of molecular sciences, 2019 - mdpi.com
Structure-based drug design is becoming an essential tool for faster and more cost-efficient
lead discovery relative to the traditional method. Genomic, proteomic, and structural studies …

Potential of quantum computing for drug discovery

Y Cao, J Romero… - IBM Journal of Research …, 2018 - ieeexplore.ieee.org
Quantum computing has rapidly advanced in recent years due to substantial development in
both hardware and algorithms. These advances are carrying quantum computers closer to …

Drugclip: Contrastive protein-molecule representation learning for virtual screening

B Gao, B Qiang, H Tan, Y Jia, M Ren… - Advances in …, 2023 - proceedings.neurips.cc
Virtual screening, which identifies potential drugs from vast compound databases to bind
with a particular protein pocket, is a critical step in AI-assisted drug discovery. Traditional …

Molecular docking and structure-based drug design strategies

LG Ferreira, RN Dos Santos, G Oliva, AD Andricopulo - Molecules, 2015 - mdpi.com
Pharmaceutical research has successfully incorporated a wealth of molecular modeling
methods, within a variety of drug discovery programs, to study complex biological and …

Role of computer-aided drug design in modern drug discovery

SJY Macalino, V Gosu, S Hong, S Choi - Archives of pharmacal research, 2015 - Springer
Drug discovery utilizes chemical biology and computational drug design approaches for the
efficient identification and optimization of lead compounds. Chemical biology is mostly …

Advancements in docking and molecular dynamics simulations towards ligand-receptor interactions and structure-function relationships

AAT Naqvi, T Mohammad, GM Hasan… - Current topics in …, 2018 - benthamdirect.com
Protein-ligand interaction is an imperative subject in structure-based drug design and
protein function prediction process. Molecular docking is a computational method which …