Bruton's kinase inhibitors for the treatment of immunological diseases: current status and perspectives

E Robak, T Robak - Journal of Clinical Medicine, 2022 - mdpi.com
The use of Bruton's tyrosine kinase (BTK) inhibitors has changed the management of
patients with B-cell lymphoid malignancies. BTK is an important molecule that interconnects …

Determinants and biomarkers of progression independent of relapses in multiple sclerosis

M Calabrese, P Preziosa, A Scalfari… - Annals of …, 2024 - Wiley Online Library
Clinical, pathological, and imaging evidence in multiple sclerosis (MS) suggests that a
smoldering inflammatory activity is present from the earliest stages of the disease and …

A review of Bruton's tyrosine kinase inhibitors in multiple sclerosis

L Airas, RA Bermel, T Chitnis… - Therapeutic …, 2024 - journals.sagepub.com
Bruton's tyrosine kinase (BTK) inhibitors are an emerging class of therapeutics in multiple
sclerosis (MS). BTK is expressed in B-cells and myeloid cells, key progenitors of which …

Antibody response to SARS-CoV-2 vaccines in patients with relapsing multiple sclerosis treated with evobrutinib: A Bruton's tyrosine kinase inhibitor

A Bar-Or, AH Cross, AL Cunningham… - Multiple Sclerosis …, 2023 - journals.sagepub.com
Background: Evobrutinib is an oral, central nervous system (CNS)-penetrant and highly
selective covalent Bruton's tyrosine kinase inhibitor under clinical development for patients …

BTK inhibition limits microglia-perpetuated CNS inflammation and promotes myelin repair

A Geladaris, S Torke, D Saberi, YB Alankus… - Acta …, 2024 - Springer
In multiple sclerosis (MS), persisting disability can occur independent of relapse activity or
development of new central nervous system (CNS) inflammatory lesions, termed chronic …

From progression to progress: The future of multiple sclerosis

J Oh, PS Giacomini, VW Yong… - Journal of Central …, 2024 - journals.sagepub.com
Significant advances have been made in the diagnosis and treatment of multiple sclerosis in
recent years yet challenges remain. The current classification of MS phenotypes according …

Efficacy and safety results after> 3.5 years of treatment with the Bruton's tyrosine kinase inhibitor evobrutinib in relapsing multiple sclerosis: Long-term follow-up of a …

X Montalban, K Piasecka-Stryczynska… - Multiple Sclerosis …, 2024 - journals.sagepub.com
Background: Evobrutinib–an oral, central nervous system (CNS)-penetrant, and highly
selective Bruton's tyrosine kinase inhibitor–has shown efficacy in a 48-week, double-blind …

Bruton's Tyrosine Kinase Inhibitors for Multiple Sclerosis Treatment: A New Frontier.

BM Greenberg - Neurologic Clinics, 2023 - europepmc.org
Multiple sclerosis (MS) can cause significant disability to patients via relapse-associated
worsening and progression independent of relapses. The causes of neuronal and myelin …

[PDF][PDF] Bruton tyrosine kinase inhibition in multiple sclerosis

LA Jayagopal, RK Zabad - Practical Neurology, 2022 - assets.bmctoday.net
30 PRACTICAL NEUROLOGY FEBRUARY 2022 lymphocytic leukemia and mantle cell
lymphoma. Despite its effectiveness for B-cell malignancies, resistance and off-target …