The energetic and allosteric landscape for KRAS inhibition

C Weng, AJ Faure, A Escobedo, B Lehner - Nature, 2024 - nature.com
Thousands of proteins have been validated genetically as therapeutic targets for human
diseases. However, very few have been successfully targeted, and many are considered …

Molecular basis of RanGTP-activated release of Histones H2A-H2B from Importin-9

JM Shaffer, J Jiou, K Tripathi, OS Olaluwoye, HYJ Fung… - Structure, 2023 - cell.com
Imp9 is the primary importin for shuttling H2A-H2B from the cytoplasm to the nucleus. It
employs an unusual mechanism where the binding of RanGTP is insufficient to release H2A …

Functional protein oligomers

S Sahoo, LR Balireddygari, AA Padhy, S Kumari… - The Three Functional …, 2025 - Elsevier
Protein oligomerization is a fundamental, yet a complex process adapted by the cell to
evolve proteins with diverse or efficient functions and enhanced stability. This evolutionary …