An overview of the synthesis and antimicrobial, antiprotozoal, and antitumor activity of thiazole and bisthiazole derivatives
Thiazole, a five-membered heteroaromatic ring, is an important scaffold of a large number of
synthetic compounds. Its diverse pharmacological activity is reflected in many clinically …
synthetic compounds. Its diverse pharmacological activity is reflected in many clinically …
A comprehensive survey upon diverse and prolific applications of chitosan-based catalytic systems in one-pot multi-component synthesis of heterocyclic rings
H Mousavi - International Journal of Biological Macromolecules, 2021 - Elsevier
Heterocyclic compounds are among the most prestigious and valuable chemical molecules
with diverse and magnificent applications in various sciences. Due to the remarkable and …
with diverse and magnificent applications in various sciences. Due to the remarkable and …
Computational bioprospecting guggulsterone against ADP ribose phosphatase of SARS-CoV-2
Coronavirus Disease-2019 (COVID-19) is a highly contagious disease caused by Severe
Acute Respiratory Syndrome-Coronavirus-2 (SARS-CoV-2). The World Health Organization …
Acute Respiratory Syndrome-Coronavirus-2 (SARS-CoV-2). The World Health Organization …
An unanticipated discovery towards novel naphthalimide corbelled aminothiazoximes as potential anti-MRSA agents and allosteric modulators for PBP2a
Available therapeutic strategies are urgently needed to conquer multidrug resistance of
MRSA. A visible effort was guided towards the advancement of novel antibacterial …
MRSA. A visible effort was guided towards the advancement of novel antibacterial …
Design, synthesis, and evaluation of antifungal bioactivity of novel pyrazole carboxamide thiazole derivatives as SDH inhibitors
M Li, W Wang, X Cheng, Y Wang, Y Chen… - Journal of Agricultural …, 2023 - ACS Publications
Agricultural production is seriously threatened by plant pathogens. The development of new
fungicides with high efficacy and low toxicity is urgently needed. In this study, a series of …
fungicides with high efficacy and low toxicity is urgently needed. In this study, a series of …
An electrochemical-enabled cascaded cyclization of enaminones with potassium thiocyanate and alcohols to access 2-alkoxythiazoles
D Li, L Chen, Y **, X Wang, L Liu, Y Li, G Chen… - Green …, 2023 - pubs.rsc.org
An electrochemical-enabled three-component cascaded cyclization of enaminones with
potassium thiocyanate and alcohols to access 2-alkoxythiazoles has been developed under …
potassium thiocyanate and alcohols to access 2-alkoxythiazoles has been developed under …
Imidazopyridine-based thiazole derivatives as potential antidiabetic agents: synthesis, in vitro bioactivity, and in silico molecular modeling approach
A new series of thiazole derivatives (4a-p) incorporating imidazopyridine moiety was
synthesized and assessed for their in vitro potential α-glucosidase potency using acarbose …
synthesized and assessed for their in vitro potential α-glucosidase potency using acarbose …
Synthesis and Biological Evaluation of Quinazolonethiazoles as New Potential Conquerors towards Pseudomonas Aeruginosa
J Wang, N Battini, MF Ansari… - Chinese Journal of …, 2021 - Wiley Online Library
Main observation and conclusion Novel quinazolonthiazoles were designed and
synthesized as new potential antimicrobial agents by facile multi‐step procedure from o …
synthesized as new potential antimicrobial agents by facile multi‐step procedure from o …
Identification of a novel antifungal backbone of naphthalimide thiazoles with synergistic potential for chemical and dynamic treatment
PL Zhang, G Lavanya, Y Yu, B Fang… - Future Medicinal …, 2021 - Taylor & Francis
Aim: The high incidence and prevalence of fungal infections call for new antifungal drugs.
This work was to develop naphthalimide thiazoles as potential antifungal agents. Results & …
This work was to develop naphthalimide thiazoles as potential antifungal agents. Results & …
[PDF][PDF] Antibacterial activity of thiazole and its derivatives
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …