[HTML][HTML] Two novel compounds, ergosterol and ergosta-5, 8-dien-3-ol, from Termitomyces heimii Natarajan demonstrate promising anti-hepatocarcinoma activity

R Ray, S Saha, S Paul - Journal of Traditional Chinese Medical Sciences, 2022 - Elsevier
Background Mushroom-derived components have immense potential to become a safe
alternative in identifying lead anti-cancer molecules. Termitomyces heimii Natarajan (T …

Identification of new inhibitors against human Great wall kinase using in silico approaches

U Ammarah, A Kumar, R Pal, NC Bal, G Misra - Scientific RepoRts, 2018 - nature.com
Microtubule associated serine/threonine kinase (MASTL) is an important Ser/Thr kinase
belonging to the family of AGC kinases. It is the human orthologue of Greatwall kinase (Gwl) …

Synthesis and in vitro study of nitro-and methoxy-2-phenylbenzofurans as human monoamine oxidase inhibitors

GL Delogu, A Kumar, G Gatto, F Bustelo… - Bioorganic …, 2021 - Elsevier
A new series of 2-phenylbenzofuran derivatives were designed and synthesized to
determine relevant structural features for the MAO inhibitory activity and selectivity. Methoxy …

New molecular scaffolds for the design of Alzheimer's acetylcholinesterase inhibitors identified using ligand-and receptor-based virtual screening

N Chitranshi, S Gupta, PK Tripathi, PK Seth - Medicinal Chemistry …, 2013 - Springer
The identification of important chemical features of acetylcholinesterase (AChE) inhibitors
will be helpful to discover the potent candidate to inhibit the AChE activity. The best …

[PDF][PDF] In Vitro screening and in silico docking analysis identifies two novel compound lecanoric acid and atranorin from Parmotrema tinctorum, exhibiting potent anti …

S Saha, R Ray, S Paul - Biointerface Res Appl Chem, 2023 - biointerfaceresearch.com
Lichens are a good repository of bio-active compounds with different pharmacological
properties; therefore, in our article, we aim to screen the antiproliferative potential of three …

Interaction between shrimp and white spot syndrome virus through PmRab7-VP28 complex: an insight using simulation and docking studies

AK Verma, S Gupta, S Verma, A Mishra… - Journal of molecular …, 2013 - Springer
White spot disease is a devastating disease of shrimp Penaeus monodon in which the
shrimp receptor protein PmRab7 interacts with viral envelop protein VP28 to form PmRab7 …

Receptor based virtual screening of potential novel inhibitors of tigar [TP53 (tumour protein 53)-induced glycolysis and apoptosis regulator

J Poyya, DJ Kumar, HG Nagendra, B Dinesh… - Medical …, 2021 - Elsevier
Abstract TP53 (tumor protein 53)-induced glycolysis and apoptosis regulator (TIGAR)
belongs to the phosphatases family of proteins that modulates the level of reactive oxygen …

Bio/chemoinformatics in India: an outlook

S Gupta, S Chavan, DN Deobagkar… - Briefings in …, 2015 - academic.oup.com
With the advent of significant establishment and development of Internet facilities and
computational infrastructure, an overview on bio/chemoinformatics is presented along with …

[PDF][PDF] In silico docking studies of alkyl esters derivative of gallic acid on Bcl-xL anti-apoptotic protein of breast cancer

RI Paramita, A Arsianti, M Radji - Int. J. Chemtech Res, 2017 - researchgate.net
Gallic acid has been reported to have various biological activities including an anticancer
effect. Numerous studies have indicated that alkyl esters derivative of gallic acid are more …

[PDF][PDF] Synthesis and cytotoxic activities of hexyl esters derivatives of gallic acid against MCF-7 cell line

RI Paramita, A Arsianti, M Radji - Oriental Journal of Chemistry, 2018 - academia.edu
Gallic acid is found in many plants, fruits, and foods where the anti-cancer activity is found.
However, gallic acid has a problem on the high polarity and low bio availability. So, it takes …