Isatin hybrids and their anti-tuberculosis activity

Z Xu, S Zhang, C Gao, J Fan, F Zhao, ZS Lv… - Chinese Chemical …, 2017‏ - Elsevier
Tuberculosis (TB) is one of the most common and even fatal infectious diseases known to
mankind. Millions of new cases are reported every year over the world, and one-third of the …

[HTML][HTML] A mini review on isatin, an anticancer scaffold with potential activities against Neglected Tropical Diseases (Ntds)

S Chowdhary, Shalini, A Arora, V Kumar - Pharmaceuticals, 2022‏ - mdpi.com
Isatin, chemically an indole-1 H-2, 3-dione, is recognised as one of the most attractive
therapeutic fragments in drug design and development. The template has turned out to be …

Indole derivatives as anti-tubercular agents: An overview on their synthesis and biological activities

GS Reddy, M Pal - Current medicinal chemistry, 2021‏ - benthamdirect.com
Background: The indole framework is considered as one of the privileged structures in the
area of medicinal chemistry and drug discovery because compounds containing this …

Transposon sequencing reveals metabolic pathways essential for Mycobacterium tuberculosis infection

AM Block, PC Wiegert, SB Namugenyi… - PLoS …, 2024‏ - journals.plos.org
New drugs are needed to shorten and simplify treatment of tuberculosis caused by
Mycobacterium tuberculosis. Metabolic pathways that M. tuberculosis requires for growth or …

Isatin derivatives with potential antitubercular activities

D Jiang, GQ Wang, X Liu, Z Zhang… - Journal of …, 2018‏ - Wiley Online Library
Tuberculosis is a life‐threatening chronic infectious disease, which primarily affects the
lungs but can spread to other vital organs. The re‐emergence and wide spread of new …

Isatin conjugates as antibacterial agents: a brief review

F Hassan, I Azad, M Asif, D Shukla, A Husain… - Medicinal …, 2023‏ - benthamdirect.com
Pathogenic bacteria, with their innate resistance to drugs, pose a constant threat to human
health and well-being and put a persistent strain on the health care system. Development of …

Mycobacterium tuberculosis chorismate mutase: A potential target for TB

M Khanapur, M Alvala, M Prabhakar, KS Kumar… - Bioorganic & medicinal …, 2017‏ - Elsevier
Mycobacterium tuberculosis chorismate mutase (Mtb CM) catalyzes the rearrangement of
chorismate to prephenate in the shikimate biosynthetic pathway to form the essential amino …

Structure–activity relationship studies of indolin‐2‐one derivatives as vascular endothelial growth factor receptor inhibitors and anticancer agents

M Yousefian, R Ghodsi - Archiv der Pharmazie, 2020‏ - Wiley Online Library
Angiogenesis is a requirement for the growth of cancer cells. The family of vascular
endothelial growth factor receptors (VEGFRs) is the main target in metastasis. Indolin‐2‐one …

Repositioning of Isatin hybrids as novel anti-tubercular agents overcoming pre-existing antibiotics resistance

R Kumar, P Takkar - Medicinal Chemistry Research, 2021‏ - Springer
The widespread deaths of tuberculosis from many decades demands an urgent need for the
development of novel anti-tubercular scaffolds that are more potent and highly selective with …

Combination of Hydrogen and Halogen Bonds in the Crystal Structures of 5-Halogeno-1H-isatin-3-oximes: Involvement of the Oxime Functionality in Halogen …

E Meier, W Seichter, M Mazik - Molecules, 2024‏ - mdpi.com
Various functional groups have been considered as acceptors for halogen bonds, but the
oxime functionality has received very little attention in this context. In this study, we focus on …