HBTM-2.1 promotes the direct asymmetric α-amination of carboxylic acids with N-aryl-N-
aroyldiazenes at low catalyst loadings (as low as 0.25 mol%), giving either 1, 3, 4-oxadiazin …

A general method for the N-arylation of amino acid esters with aryl triflates is described. Both
α-and β-amino acid esters, including methyl, tert-butyl, and benzyl esters, are viable …

Fe3O4@ SiO2 nanoparticles was functionalized with a binuclear Schiff base Cu (II)‐complex
(Fe3O4@ SiO2/Schiff base‐Cu (II) NPs) and used as an effective magnetic hetereogeneous …

Different cross-coupling reactions for the formation of biologically important motifs and
intermediates in organic synthesis using various suitable copper catalysts are reviewed …

Polypeptides present remarkable selectivity challenges for chemical methods. Amino groups
are ubiquitous in polypeptide structure, yet few paradigms exist for reactivity and selectivity …

Impact of microwave radiation on organic chemistry has been assessed by workers time to
time. This review covers selected recent examples form cross-coupling reactions …

A mild and efficient method for the N-arylation of zwitterionic amino acids, amino acid esters
and peptides is described. The procedure provides the first room temperature synthesis of N …

N-Arylation of carbazole has been achieved in high yields within 1 h using a microwave-
assisted catalytic CuI reaction with no organic ligand. The N-arylation can be performed by …

A robust, mild, and efficient method for the Pd‐catalyzed N‐heteroarylation of optically pure
α‐amino esters was developed. Dichloro [1, 3‐bis (2, 6‐di‐3‐pentylphenyl) imidazol‐2 …

In the last decade, our group has been very active at develo** and assaying complex
libraries of scaffolds with a focus on their potential to identify bioactive drug candidates for …