Discovery of PIM-1 kinase inhibitors based on the 2, 5-disubstituted 1, 3, 4-oxadiazole scaffold against prostate cancer: Design, synthesis, in vitro and in vivo …

AS Castanet, MS Nafie, SA Said, RK Arafa - European Journal of Medicinal …, 2023‏ - Elsevier
PIM-1 kinases play an established role in prostate cancer development and progression.
This research work tackles the design and synthesis of new PIM-1 kinase targeting 2, 5 …

Design, synthesis, and biological evaluation of novel psoralen-based 1, 3, 4-oxadiazoles as potent fungicide candidates targeting pyruvate kinase

J Dong, W Gao, K Li, Z Hong, L Tang… - Journal of Agricultural …, 2022‏ - ACS Publications
Pyruvate kinase (PK) has been considered as a promising fungicide target discovered in our
previous studies. Natural compounds are important sources for discovery and development …

Design, synthesis, and evaluation of antitumor activity in Pseudolaric acid B azole derivatives: Novel and potent angiogenesis inhibitor via regulation of the PI3K/AKT …

H Deng, Q Xu, XT Li, X Huang, JY Liu, R Yan… - European Journal of …, 2024‏ - Elsevier
Tumor proliferation and metastasis are intricately linked to blood vessel formation, with
vascular endothelial growth factor (VEGF) playing a pivotal role in orchestrating …

Anti-cancer activity of capsaicin and its analogs in gynecological cancers

KC Brown, AM Sugrue, KB Conley… - … in cancer research, 2024‏ - pubmed.ncbi.nlm.nih.gov
Capsaicin is the hot and pungent ingredient of chili peppers. It is a potent pain-relieving
agent and is often present in over-the-counter analgesic lotions and creams. Several …

1, 2, 3-Triazole tethered hybrid capsaicinoids as antiproliferative agents active against lung cancer cells (A549)

A Khan, F Naaz, R Basit, D Das, P Bisht, M Shaikh… - ACS …, 2022‏ - ACS Publications
A series of novel 1, 2, 3-triazole derivatives of capsaicin and its structural isomer (new
natural product hybrid capsaicinoid) were synthesized by exploiting one-/two-point …

[HTML][HTML] Synthesis and Cytotoxic Activity of 1,2,4-Triazolo-Linked Bis-Indolyl Conjugates as Dual Inhibitors of Tankyrase and PI3K

PA Yakkala, SR Panda, S Shafi, VGM Naidu, MS Yar… - Molecules, 2022‏ - mdpi.com
A series of new 1, 2, 4-triazolo-linked bis-indolyl conjugates (15a–r) were prepared by
multistep synthesis and evaluated for their cytotoxic activity against various human cancer …

Capsaicin derivatives: Synthesis and biological activity

S Liu, X Zheng, J Wu, Y Zeng, X Wei… - Chemical Biology & …, 2024‏ - Wiley Online Library
Capsaicin is the main active ingredient of chili peppers and the most pungent alkaloid. It is
reported that capsaicin has many pharmacological effects such as analgesia, anticancer …

Interlinking Human-Derived Leukemia Cells with Clinicopathological Therapeutics: Exploring Capsaicin's Anti-Cancer Mechanisms/potential for Leukemia Patients …

M Mastoor, F Choudhry, A Khurshid… - Pakistan Journal of …, 2024‏ - mail.thejas.com.pk
Capsaicin, a bioactive compound isolated from chilli peppers, comes out as a potential
agent for its anti-proliferation role in leukemia patients' therapy. Objectives: This systematic …