Thiazole ring—A biologically active scaffold
A Petrou, M Fesatidou, A Geronikaki - Molecules, 2021 - mdpi.com
Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical
applications. Its derivatives have a wide range of biological activities such as antioxidant …
applications. Its derivatives have a wide range of biological activities such as antioxidant …
Development and therapeutic potential of 2-aminothiazole derivatives in anticancer drug discovery
Currently, the development of anticancer drug resistance is significantly restricted the clinical
efficacy of the most commonly prescribed anticancer drug. Malignant disease is widely …
efficacy of the most commonly prescribed anticancer drug. Malignant disease is widely …
A retrospect on antimicrobial potential of thiazole scaffold
Due to its appreciable diversity in biological actions, thiazole and its substituted
components, a significant class of heterocyclic compounds has developed as an influential …
components, a significant class of heterocyclic compounds has developed as an influential …
Anticancer potential of thiazole derivatives: a retrospective review
S Jain, S Pattnaik, K Pathak, S Kumar… - Mini reviews in …, 2018 - ingentaconnect.com
This review brings forth the potential of thiazole derivatives for their anticancer activities. The
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
[PDF][PDF] Antibacterial activity of thiazole and its derivatives
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
Heterocycle compounds with antimicrobial activity
M Fesatidou, A Petrou, G Athina - Current pharmaceutical …, 2020 - ingentaconnect.com
Background: Bacterial infections are a growing problem worldwide causing morbidity and
mortality mainly in develo** countries. Moreover, the increased number of …
mortality mainly in develo** countries. Moreover, the increased number of …
Review on synthetic chemistry and antibacterial importance of thiazole derivatives
Background: Thiazole is one of the leading heterocyclic five-member ring compounds that
contain nitrogen and sulphur atom. Many natural and/or synthetic compounds contain …
contain nitrogen and sulphur atom. Many natural and/or synthetic compounds contain …
2, 4-Disubstituted thiazoles as multitargated bioactive molecules
Thiazoles are important heterocyclics exhibiting boundaryless biological activities, such as
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …
Synthesis, in silico and biological studies of thiazolyl-2h-chromen-2-one derivatives as potent antitubercular agents
BS Jadhav, RS Yamgar, RS Kenny… - … -Aided Drug Design, 2020 - ingentaconnect.com
Background: A series of new six thiazolyl-2-amine-based Schiff base derivatives (4a-4f)
were synthesized by a sequential multistep reaction starting with Salicylaldehyde. Methods …
were synthesized by a sequential multistep reaction starting with Salicylaldehyde. Methods …
[HTML][HTML] Quorum sensing inhibitors: curbing pathogenic infections through inhibition of bacterial communication
Currently, most of the developed and develo** countries are facing the problem of
infectious diseases. The genius way of an exaggerated application of antibiotics led the …
infectious diseases. The genius way of an exaggerated application of antibiotics led the …