Metalloproteinases and their inhibitors: potential for the development of new therapeutics

M Raeeszadeh-Sarmazdeh, LD Do, BG Hritz - Cells, 2020 - mdpi.com
The metalloproteinase (MP) family of zinc-dependent proteases, including matrix
metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs), and a disintegrin …

Missing the target: matrix metalloproteinase antitargets in inflammation and cancer

A Dufour, CM Overall - Trends in pharmacological sciences, 2013 - cell.com
Matrix metalloproteinases (MMPs) are reputed to cause the inflammatory tissue destruction
characterizing chronic inflammatory diseases and to degrade basement membrane …

Therapeutic potential of matrix metalloproteinase inhibition in breast cancer

ES Radisky… - Journal of cellular …, 2017 - Wiley Online Library
Matrix metalloproteinases (MMPs) are a family of zinc endopeptidases that cleave nearly all
components of the extracellular matrix as well as many other soluble and cell‐associated …

Selective inhibitors of medium-size S1′ pocket matrix metalloproteinases: a step** stone of future drug discovery

SK Baidya, S Banerjee, N Adhikari… - Journal of Medicinal …, 2022 - ACS Publications
Among various matrix metalloproteinases (MMPs), MMPs having medium-size S1′ pockets
are established as promising biomolecular targets for executing crucial roles in cancer …

[HTML][HTML] Matrix metalloproteinases as breast cancer drivers and therapeutic targets

ES Radisky, DC Radisky - Frontiers in bioscience (Landmark …, 2015 - ncbi.nlm.nih.gov
Members of the matrix metalloproteinase (MMP) family have been identified as poor
prognosis markers for breast cancer patients and as drivers of many facets of the tumor …

Extracellular matrix: emerging roles and potential therapeutic targets for breast cancer

Y Zhao, X Zheng, Y Zheng, Y Chen, W Fei… - Frontiers in …, 2021 - frontiersin.org
Increasing evidence shows that the extracellular matrix (ECM) is an important regulator of
breast cancer (BC). The ECM comprises of highly variable and dynamic components …

Matrix metalloproteinases as new targets in Alzheimer's disease: Opportunities and challenges

P Zipfel, C Rochais, K Baranger, S Rivera… - Journal of Medicinal …, 2020 - ACS Publications
Although matrix metalloproteinases (MMPs) are implicated in the regulation of numerous
physiological processes, evidence of their pathological roles have also been obtained in the …

Assessing structural insights into in-house arylsulfonyl L-(+) glutamine MMP-2 inhibitors as promising anticancer agents through structure-based computational …

SK Baidya, S Banerjee, B Ghosh, T Jha… - SAR and QSAR in …, 2023 - Taylor & Francis
ABSTRACT MMP-2 is potentially contributing to several cancer progressions including
leukaemias. Therefore, considering MMP-2 as a promising target, novel anticancer …

C-terminal truncation of IFN-γ inhibits proinflammatory macrophage responses and is deficient in autoimmune disease

A Dufour, CL Bellac, U Eckhard, N Solis, T Klein… - Nature …, 2018 - nature.com
Controlled macrophage differentiation and activation in the initiation and resolution of
inflammation is crucial for averting progression to chronic inflammatory and autoimmune …

[HTML][HTML] Regulation and involvement of matrix metalloproteinases in vascular diseases

M Amin, S Pushpakumar, N Muradashvili… - Frontiers in …, 2016 - ncbi.nlm.nih.gov
Matrix metalloproteinases (MMPs) are a family of zinc dependent endopeptidases whose
main function is to degrade and deposit structural proteins within the extracellular matrix …