Isoxazolidine: a privileged scaffold for organic and medicinal chemistry
M Berthet, T Cheviet, G Dujardin, I Parrot… - Chemical …, 2016 - ACS Publications
The isoxazolidine ring represents one of the privileged structures in medicinal chemistry,
and there have been an increasing number of studies on isoxazolidine and isoxazolidine …
and there have been an increasing number of studies on isoxazolidine and isoxazolidine …
Recent advances in indium-promoted organic reactions
J Auge, N Lubin-Germain, J Uziel - Synthesis, 2007 - thieme-connect.com
This review deals with organic reactions which are promoted by indium metal or indium
salts, with a focus on recent advances in stoichiometric and catalytic pathways. Applications …
salts, with a focus on recent advances in stoichiometric and catalytic pathways. Applications …
Cp∗ Ir-catalyzed N-alkylation of amines with alcohols. A versatile and atom economical method for the synthesis of amines
K Fujita, Y Enoki, R Yamaguchi - Tetrahedron, 2008 - Elsevier
A versatile and highly atom economical catalytic system consisting of [Cp∗ IrCl2] 2/NaHCO3
(Cp∗= pentamethylcyclopentadienyl) for the N-alkylation of amines with primary and …
(Cp∗= pentamethylcyclopentadienyl) for the N-alkylation of amines with primary and …
Dual catalysis for enantioselective convergent synthesis of enantiopure vicinal amino alcohols
Enantiopure vicinal amino alcohols and derivatives are essential structural motifs in natural
products and pharmaceutically active molecules, and serve as main chiral sources in …
products and pharmaceutically active molecules, and serve as main chiral sources in …
Metal‐Free Reductive Cleavage of C N and S N Bonds by Photoactivated Electron Transfer from a Neutral Organic Donor
A photoactivated neutral organic super electron donor cleaves challenging
arenesulfonamides derived from dialkylamines at room temperature. It also cleaves a) ArC …
arenesulfonamides derived from dialkylamines at room temperature. It also cleaves a) ArC …
Harnessing phosphonate antibiotics argolaphos biosynthesis enables a synthetic biology-based green synthesis of glyphosate
L Chu, X Luo, T Zhu, Y Cao, L Zhang, Z Deng… - Nature …, 2022 - nature.com
Glyphosate is a widely used herbicide with an annual production of more than one million
tons globally. Current commercialized production processes of glyphosate are generally …
tons globally. Current commercialized production processes of glyphosate are generally …
Radical cation and neutral radical of aza-thia [7] helicene with SOMO–HOMO energy level inversion
Y Wang, H Zhang, M Pink, A Olankitwanit… - Journal of the …, 2016 - ACS Publications
We report a relatively persistent, open-shell aza-thia [7] helicene with cross-conjugated
electron-rich π-system. The singly occupied molecular orbital (SOMO) energy levels of both …
electron-rich π-system. The singly occupied molecular orbital (SOMO) energy levels of both …
Total synthesis of (±)-haouamine A
The first total synthesis of the highly complex and potent anticancer agent haouamine A is
reported through an eight-step sequence. Brevity of the sequence and complete control of …
reported through an eight-step sequence. Brevity of the sequence and complete control of …
Intermolecular Cope-type hydroamination of alkenes and alkynes using hydroxylamines
The development of the Cope-type hydroamination as a method for the metal-and acid-free
intermolecular hydroamination of hydroxylamines with alkenes and alkynes is described …
intermolecular hydroamination of hydroxylamines with alkenes and alkynes is described …
Stereoselective isoxazolidine synthesis via copper-catalyzed alkene aminooxygenation
Isoxazolidines are useful in organic synthesis, drug discovery, and chemical biology
endeavors. A new stereoselective synthesis of methyleneoxy-substituted isoxazolidines is …
endeavors. A new stereoselective synthesis of methyleneoxy-substituted isoxazolidines is …