[HTML][HTML] Glucagon-like peptide-1 receptor co-agonists for treating metabolic disease

LL Baggio, DJ Drucker - Molecular metabolism, 2021‏ - Elsevier
Background Glucagon-like peptide-1 receptor (GLP-1R) agonists are approved for the
treatment of type 2 diabetes and obesity and elicit robust improvements in glycemic control …

[HTML][HTML] Glucagon-like peptide-1 (GLP-1) receptor agonists and neuroinflammation: Implications for neurodegenerative disease treatment

KO Kopp, EJ Glotfelty, Y Li, NH Greig - Pharmacological research, 2022‏ - Elsevier
Chronic, excessive neuroinflammation is a key feature of neurodegenerative diseases such
as Alzheimer's disease (AD) and Parkinson's disease (PD). However, neuroinflammatory …

[HTML][HTML] Effects on weight loss and glycemic control with SAR441255, a potent unimolecular peptide GLP-1/GIP/GCG receptor triagonist

M Bossart, M Wagner, R Elvert, A Evers, T Hübschle… - Cell metabolism, 2022‏ - cell.com
Unimolecular triple incretins, combining the activity of glucagon-like peptide-1 (GLP-1),
glucose-dependent insulinotropic polypeptide (GIP), and glucagon (GCG), have …

Incretin hormones: Their role in health and disease

MA Nauck, JJ Meier - Diabetes, Obesity and Metabolism, 2018‏ - Wiley Online Library
Incretin hormones are gut peptides that are secreted after nutrient intake and stimulate
insulin secretion together with hyperglycaemia. GIP (glucose‐dependent insulinotropic …

GIP as a therapeutic target in diabetes and obesity: insight from incretin co-agonists

JJ Holst, MM Rosenkilde - The Journal of Clinical Endocrinology …, 2020‏ - academic.oup.com
The 2 hormones responsible for the amplification of insulin secretion after oral as opposed
to intravenous nutrient administration are the gut peptides, glucagon-like peptide-1 (GLP-1) …

Separate and combined glucometabolic effects of endogenous glucose-dependent insulinotropic polypeptide and glucagon-like peptide 1 in healthy individuals

LS Gasbjerg, MM Helsted, B Hartmann, MH Jensen… - Diabetes, 2019‏ - Am Diabetes Assoc
The incretin hormones glucose-dependent insulinotropic polypeptide (GIP) and glucagon-
like peptide 1 (GLP-1) are secreted postprandially and contribute importantly to postprandial …

Evaluation of the incretin effect in humans using GIP and GLP-1 receptor antagonists

LS Gasbjerg, NC Bergmann, S Stensen… - Peptides, 2020‏ - Elsevier
Glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1)
potentiate glucose-induced insulin secretion and are therefore thought to be responsible for …

GLP-1 receptor agonist treatment increases bone formation and prevents bone loss in weight-reduced obese women

EW Iepsen, JR Lundgren, B Hartmann… - The Journal of …, 2015‏ - academic.oup.com
Context: Recent studies indicate that glucagon-like peptide (GLP)-1 regulates bone
turnover, but the effects of GLP-1 receptor agonists (GLP-1 RAs) on bone in obese weight …

Gut hormones and their effect on bone metabolism. Potential drug therapies in future osteoporosis treatment

SP Schiellerup, K Skov-Jeppesen… - Frontiers in …, 2019‏ - frontiersin.org
Bone homeostasis displays a circadian rhythm with increased resorption during the night
time as compared to day time, a difference that seems—at least partly—to be caused by food …

The associations of gut microbiota, endocrine system and bone metabolism

Y Tu, X Kuang, L Zhang, X Xu - Frontiers in Microbiology, 2023‏ - frontiersin.org
Gut microbiota is of great importance in human health, and its roles in the maintenance of
skeletal homeostasis have long been recognized as the “gut-bone axis.” Recent evidence …