The indole alkaloids, ranging from lysergic acid to vincristine, have long inspired organic
synthesis chemists. Interest in develo** new methods for indole synthesis has burgeoned …

Natural product synthesis is a highly demanding field in constant need of efficient
transformations that allow either straightforward, scalable, and high-yielding preparation of …

The C–N cross-coupling chemistry intensely developed since the late 1990s has supplied
synthesists with an overwhelming number of methods to effectively combine carbon and …

This perspective reports on some of the main copper-catalyzed routes to the construction of
the pyrrole and furan rings incorporated into the indole and benzo [b] furan systems …

Copper-catalyzed cross-coupling reactions which lead to the formation of C–N, C–O, C–S
and C–C bonds have been recognized as one of the most useful strategies in synthetic …

Published data of the last 10 years concerning the development of new and upgrading of
known approaches to indole synthesis are integrated and analyzed. Modern versions of the …

A regioselective synthesis of indole‐3‐carboxylic acid esters from anilines and diazo
compounds has been realized by making use of the pyrimidyl group‐assisted rhodium …

Multisubstituted indoles were synthesized via a one-pot tandem copper-catalyzed Ullmann-
type C–N bond formation/intramolecular cross-dehydrogenative coupling process at 130° C …

We herein describe a palladium-catalyzed formal aromaticity transfer coupling reaction
between phenols and pyrrolidines or indolines to generate the corresponding N-cyclohexyl …

Background: Due to significant biological activity associated with N-, O-and S-heterocycles,
a number of reports for their synthesis have appeared in recent decades. Traditional …