The PI3K-Akt-mTOR signaling pathway in human acute myeloid leukemia (AML) cells

I Nepstad, KJ Hatfield, IS Grønningsæter… - International journal of …, 2020‏ - mdpi.com
Acute myeloid leukemia (AML) is a heterogeneous group of diseases characterized by
uncontrolled proliferation of hematopoietic stem cells in the bone marrow. Malignant cell …

PI3K signaling in cancer: beyond AKT

EC Lien, CC Dibble, A Toker - Current opinion in cell biology, 2017‏ - Elsevier
The phosphoinositide 3-kinase (PI3K) signaling pathway is one of the most frequently
altered pathways in human cancer and has a critical role in driving tumor initiation and …

PI3K/Akt/mTOR and Ras/Raf/MEK/ERK signaling pathways inhibitors as anticancer agents: Structural and pharmacological perspectives

V Asati, DK Mahapatra, SK Bharti - European journal of medicinal chemistry, 2016‏ - Elsevier
The protein kinases regulate cellular functions such as transcription, translation,
proliferation, growth and survival by the process of phosphorylation. Over activation of …

New concepts and mechanisms of platelet activation signaling

B Estevez, X Du - Physiology, 2017‏ - journals.physiology.org
Upon blood vessel injury, platelets are exposed to adhesive proteins in the vascular wall
and soluble agonists, which initiate platelet activation, leading to formation of hemostatic …

Epithelial-to-mesenchymal transition is a cause of both intrinsic and acquired resistance to KRAS G12C inhibitor in KRAS G12C–mutant non–small cell lung cancer

Y Adachi, K Ito, Y Hayashi, R Kimura… - Clinical Cancer …, 2020‏ - aacrjournals.org
Purpose: KRAS is among the most commonly mutated oncogene in cancer including non–
small cell lung cancer (NSCLC). In early clinical trials, inhibitors targeting G12C-mutant …

Dual or multi-targeting inhibitors: The next generation anticancer agents

NM Raghavendra, D **ili, S Kadasi, A Mettu… - European journal of …, 2018‏ - Elsevier
Dual-targeting/Multi-targeting of oncoproteins by a single drug molecule represents an
efficient, logical and alternative approach to drug combinations. An increasing interest in this …

Molecular distinction between physiological and pathological cardiac hypertrophy: experimental findings and therapeutic strategies

BC Bernardo, KL Weeks, L Pretorius… - Pharmacology & …, 2010‏ - Elsevier
Cardiac hypertrophy can be defined as an increase in heart mass. Pathological cardiac
hypertrophy (heart growth that occurs in settings of disease, eg hypertension) is a key risk …

Molecular and cellular pathways contributing to brain aging

A Zia, AM Pourbagher-Shahri, T Farkhondeh… - Behavioral and Brain …, 2021‏ - Springer
Aging is the leading risk factor for several age-associated diseases such as
neurodegenerative diseases. Understanding the biology of aging mechanisms is essential …

PIK3CA in cancer: The past 30 years

R Arafeh, Y Samuels - Seminars in cancer biology, 2019‏ - Elsevier
Almost thirty years ago, PI3K was discovered as a lipid kinase associated with certain
oncoproteins. The first decade of research on PI3K saw the identification, purification and …

PI3K-Akt pathway: its functions and alterations in human cancer

M Osaki, M Oshimura, H Ito - Apoptosis, 2004‏ - Springer
Abstract Phosphatidylinositol-3-kinase (PI3K) is a lipid kinase and generates
phosphatidylinositol-3, 4, 5-trisphosphate (PI (3, 4, 5) P3). PI (3, 4, 5) P3 is a second …