Advances of artificial intelligence in anti-cancer drug design: a review of the past decade

L Wang, Y Song, H Wang, X Zhang, M Wang, J He… - Pharmaceuticals, 2023 - mdpi.com
Anti-cancer drug design has been acknowledged as a complicated, expensive, time-
consuming, and challenging task. How to reduce the research costs and speed up the …

Sequence-based drug design as a concept in computational drug design

L Chen, Z Fan, J Chang, R Yang, H Hou, H Guo… - Nature …, 2023 - nature.com
Drug development based on target proteins has been a successful approach in recent
decades. However, the conventional structure-based drug design (SBDD) pipeline is a …

The changing scenario of drug discovery using AI to deep learning: Recent advancement, success stories, collaborations, and challenges

C Chakraborty, M Bhattacharya, SS Lee… - Molecular Therapy …, 2024 - pmc.ncbi.nlm.nih.gov
Due to the transformation of artificial intelligence (AI) tools and technologies, AI-driven drug
discovery has come to the forefront. It reduces the time and expenditure. Due to these …

Geometric interaction graph neural network for predicting protein–ligand binding affinities from 3d structures (gign)

Z Yang, W Zhong, Q Lv, T Dong… - The journal of physical …, 2023 - ACS Publications
Predicting protein–ligand binding affinities (PLAs) is a core problem in drug discovery.
Recent advances have shown great potential in applying machine learning (ML) for PLA …

Learning size-adaptive molecular substructures for explainable drug–drug interaction prediction by substructure-aware graph neural network

Z Yang, W Zhong, Q Lv, CYC Chen - Chemical science, 2022 - pubs.rsc.org
Drug–drug interactions (DDIs) can trigger unexpected pharmacological effects on the body,
and the causal mechanisms are often unknown. Graph neural networks (GNNs) have been …

Drug–target binding affinity prediction model based on multi-scale diffusion and interactive learning

Z Zhu, X Zheng, G Qi, Y Gong, Y Li, N Mazur… - Expert Systems with …, 2024 - Elsevier
Drug–target interactions (DTIs) play a key role in drug discovery and development as they
are critical in understanding the complex mechanisms of underlying drugs and their …

MGraphDTA: deep multiscale graph neural network for explainable drug–target binding affinity prediction

Z Yang, W Zhong, L Zhao, CYC Chen - Chemical science, 2022 - pubs.rsc.org
Predicting drug–target affinity (DTA) is beneficial for accelerating drug discovery. Graph
neural networks (GNNs) have been widely used in DTA prediction. However, existing …

DeepMGT-DTI: Transformer network incorporating multilayer graph information for Drug–Target interaction prediction

P Zhang, Z Wei, C Che, B ** - Computers in biology and medicine, 2022 - Elsevier
Drug–target interaction (DTI) prediction reduces the cost and time of drug development, and
plays a vital role in drug discovery. However, most of research does not fully explore the …

Meta learning with graph attention networks for low-data drug discovery

Q Lv, G Chen, Z Yang, W Zhong… - IEEE Transactions on …, 2023 - ieeexplore.ieee.org
Finding candidate molecules with favorable pharmacological activity, low toxicity, and
proper pharmacokinetic properties is an important task in drug discovery. Deep neural …

AttentionMGT-DTA: A multi-modal drug-target affinity prediction using graph transformer and attention mechanism

H Wu, J Liu, T Jiang, Q Zou, S Qi, Z Cui, P Tiwari… - Neural Networks, 2024 - Elsevier
The accurate prediction of drug-target affinity (DTA) is a crucial step in drug discovery and
design. Traditional experiments are very expensive and time-consuming. Recently, deep …