Understanding and overcoming resistance to PARP inhibitors in cancer therapy

MP Dias, SC Moser, S Ganesan… - Nature reviews Clinical …, 2021 - nature.com
Develo** novel targeted anticancer therapies is a major goal of current research. The use
of poly (ADP-ribose) polymerase (PARP) inhibitors in patients with homologous …

[HTML][HTML] DNA damage response in cancer therapy and resistance: challenges and opportunities

D Jurkovicova, CM Neophytou, AČ Gašparović… - International Journal of …, 2022 - mdpi.com
Resistance to chemo-and radiotherapy is a common event among cancer patients and a
reason why new cancer therapies and therapeutic strategies need to be in continuous …

[HTML][HTML] Vorinostat (SAHA) and breast cancer: an overview

A Wawruszak, L Borkiewicz, E Okon, W Kukula-Koch… - Cancers, 2021 - mdpi.com
Simple Summary Breast cancer (BC) is the most frequent malignancy diagnosed in 2020
worldwide. Despite significant advances in BC therapy, its pathogenesis is still not fully …

New approaches in breast cancer therapy through green nanotechnology and nano-ayurvedic medicine–pre-clinical and pilot human clinical investigations

M Khoobchandani, KK Katti… - International journal …, 2020 - Taylor & Francis
Purpose The overarching objective of this investigation was to investigate the intervention of
green nanotechnology to transform the ancient holistic Ayurvedic medicine scientifically …

[HTML][HTML] PARP1: Structural insights and pharmacological targets for inhibition

JO Spiegel, B Van Houten, JD Durrant - DNA repair, 2021 - Elsevier
Abstract Poly (ADP-ribose) polymerase 1 (PARP1, also known as ADPRT1) is a
multifunctional human ADP-ribosyltransferase. It plays a role in multiple DNA repair …

Platinum-based systematic therapy in triple-negative breast cancer

Y Zhu, Y Hu, C Tang, X Guan, W Zhang - Biochimica et Biophysica Acta …, 2022 - Elsevier
Due to the lack of definitive hormone receptors, triple negative breast cancer (TNBC)
patients receive little clinical benefit from endocrine or molecular targeted therapies, leading …

Inhibition of histone deacetylases attenuates tumor progression and improves immunotherapy in breast cancer

B Lian, X Chen, K Shen - Frontiers in Immunology, 2023 - frontiersin.org
Breast cancer is one of the common malignancies with poor prognosis worldwide. The
treatment of breast cancer patients includes surgery, radiation, hormone therapy …

[HTML][HTML] Proteins from the DNA damage response: Regulation, dysfunction, and anticancer strategies

C Molinaro, A Martoriati, K Cailliau - Cancers, 2021 - mdpi.com
Simple Summary Cells respond to genotoxic stress through complex protein pathways
called DNA damage response (DDR). These mechanisms ensure the preservation of …

Exploring the potential of metallodrugs as chemotherapeutics for triple negative breast cancer

N Nayeem, M Contel - Chemistry–A European Journal, 2021 - Wiley Online Library
This review focuses on studies of coordination and organometallic compounds as potential
chemotherapeutics against triple negative breast cancer (TNBC) which has one of the …

Selective PARP1 inhibitors, PARP1-based dual-target inhibitors, PROTAC PARP1 degraders, and prodrugs of PARP1 inhibitors for cancer therapy

X Peng, W Pan, F Jiang, W Chen, Z Qi, W Peng… - Pharmacological …, 2022 - Elsevier
Poly ADP-ribose polymerase (PARP) plays a critical role in many cellular processes such as
DNA damage repair, gene transcription and cell apoptosis. Therefore, targeting PARP …