Synthesis, antimicrobial activity, and molecular modeling studies of some benzoxazole derivatives

MT Muhammed, G Kuyucuklu… - Letters in Drug …, 2022 - ingentaconnect.com
Background: The need to develop novel antimicrobial agents is apparent as infectious
diseases are increasing and resistance is rapidly develo** against the drugs used in the …

Design, synthesis, molecular docking, density functional theory and antimicrobial studies of some novel benzoxazole derivatives as structural bioisosteres of …

M Erol, I Celik, O Temiz-Arpaci… - Journal of …, 2021 - Taylor & Francis
A series of some novel 2-(p-tert-butylphenyl)-5-(3-substituted-propionamido) benzoxazole
derivatives have been designed, synthesized, evaluated for antimicrobial activity and have …

Synthesis, antimicrobial activity, density functional modelling and molecular docking with COVID-19 main protease studies of benzoxazole derivative: 2-(p-chloro …

CT Zeyrek, ÖT Arpacı, M Arısoy, FK Onurdağ - Journal of Molecular …, 2021 - Elsevier
This study contains synthesis, antimicrobial activity, density functional modelling and
molecular docking studies of benzoxazole derivative: 2-(p-chloro-benzyl)-5-[3-(4-ethly-1 …

Synthesis, molecular docking, and DFT studies of some new 2, 5-disubstituted benzoxazoles as potential antimicrobial and cytotoxic agents

M Erol, I Celik, E Uzunhisarcikli… - Polycyclic Aromatic …, 2022 - Taylor & Francis
In this study, a total of 17 piece 2, 5-disubstituted benzoxazole derivatives were synthesized,
2 of which were not original, their antimicrobial activities were determined using …

Synthesis, quantum mechanical calculations, antimicrobial activities and molecular docking studies of five novel 2, 5-disubstituted benzoxazole derivatives

O Temiz-Arpaci, CT Zeyrek, M Arisoy, M Erol… - Journal of Molecular …, 2021 - Elsevier
In this study, five new 2-(p-(Substituted) phenyl)-5-(3-(4-ethylpiperazine-1-yl) propionamido)
benzoxazole derivatives (B7-B11) were designed, synthesized, and their antimicrobial …

In Vitro and In Silico Studies of Quinoline-2-Carbaldehyde Hydrazone Derivatives as Potent Antimicrobial Agents

I Celik, M Erol, MO Puskullu… - Polycyclic Aromatic …, 2022 - Taylor & Francis
We previously synthesized a series of quinoline-2-carbaldehyde hydrazone derivatives and
evaluated their antioxidant activities. In this study, the antimicrobial activities of these …

Synthesis, molecular structure and biological activity of Niii complexes based on substituted 2-(2-hydroxyphenyl) benzoxazole

IO Tupaeva, OP Demidov, EV Vetrova… - Mendeleev …, 2022 - Elsevier
New Ni ii complexes based on the substituted 2-(2-hydroxy-phenyl) benzoxazole have been
synthesized from the corresponding ligands and nickel acetate. The crystal structure of bis [2 …

[PDF][PDF] In vitro haemolytic, antioxidant and antibacterial (ESBLs and MRSA) activity of Datura metel L. flower and leaf extracts

P Srinivasan, MSR Inala, N HS - 2021 - nopr.niscpr.res.in
Prevalence of antibiotic resistant bacteria is an issue of concern as it affects the efficiency of
antibiotics significantly. It makes the drug manufacturers continuously search for newer …

[PDF][PDF] Synthesis, antimicrobial and in silico studies of new 2.5-disubstituted benzoxazole derivative

M Erol, I Celik, G Kuyucuklu - Med. Sci. Int. Med. J, 2021 - manage.effectpublishing.com
In this study, a new 2.5-substituted benzoxazole derivative compound was synthesized in
three steps, its antimicrobial activities were determined by the microdilution method on …

Synthesis of some new benzoxazole derivatives and antimicrobial and cytotoxic activity studies

M Erol, İ Çelik, G Kuyucuklu… - Avrupa Bilim ve Teknoloji …, 2021 - dergipark.org.tr
There is an urgent need to develop new antimicrobial drugs due to the rapid development of
resistance to increasing microbial infectious diseases and drugs used in their treatment …