[HTML][HTML] Sirtuin signaling in cellular senescence and aging

SH Lee, JH Lee, HY Lee, KJ Min - BMB reports, 2019 - ncbi.nlm.nih.gov
Sirtuin is an essential factor that delays cellular senescence and extends the organismal
lifespan through the regulation of diverse cellular processes. Suppression of cellular …

Sirtuin activators and inhibitors: Promises, achievements, and challenges

H Dai, DA Sinclair, JL Ellis, C Steegborn - Pharmacology & therapeutics, 2018 - Elsevier
The NAD+-dependent protein lysine deacylases of the Sirtuin family regulate various
physiological functions, from energy metabolism to stress responses. The human Sirtuin …

Pyridinium salts: from synthesis to reactivity and applications

S Sowmiah, JMSS Esperança, LPN Rebelo… - Organic Chemistry …, 2018 - pubs.rsc.org
Structurally diverse pyridinium salts are quite familiar structures in many natural products
and bioactive pharmaceuticals. Over the centuries, these privileged scaffolds have played …

Sirtuin functions and modulation: from chemistry to the clinic

V Carafa, D Rotili, M Forgione, F Cuomo… - Clinical …, 2016 - Springer
Sirtuins are NAD+-dependent histone deacetylases regulating important metabolic
pathways in prokaryotes and eukaryotes and are involved in many biological processes …

Mitochondrial dysfunction in the pathophysiology of renal diseases

R Che, Y Yuan, S Huang… - American Journal of …, 2014 - journals.physiology.org
Mitochondrial dysfunction has gained recognition as a contributing factor in many diseases.
The kidney is a kind of organ with high energy demand, rich in mitochondria. As such …

Seven sirtuins for seven deadly diseases ofaging

BJ Morris - Free Radical Biology and Medicine, 2013 - Elsevier
Sirtuins are a class of NAD+-dependent deacetylases having beneficial health effects. This
extensive review describes the numerous intracellular actions of the seven mammalian …

Pharmacological approaches to restore mitochondrial function

PA Andreux, RH Houtkooper, J Auwerx - Nature reviews Drug …, 2013 - nature.com
Mitochondrial dysfunction is not only a hallmark of rare inherited mitochondrial disorders but
also implicated in age-related diseases, including those that affect the metabolic and …

Sirtuin activators and inhibitors

JM Villalba, FJ Alcaín - Biofactors, 2012 - Wiley Online Library
Abstract Sirtuins 1‐7 (SIRT1‐7) belong to the third class of deacetylase enzymes, which are
dependent on NAD+ for activity. Sirtuins activity is linked to gene repression, metabolic …

Ex-527 inhibits Sirtuins by exploiting their unique NAD+-dependent deacetylation mechanism

M Gertz, F Fischer, GTT Nguyen… - Proceedings of the …, 2013 - National Acad Sciences
Sirtuins are protein deacetylases regulating metabolism and stress responses. The seven
human Sirtuins (Sirt1–7) are attractive drug targets, but Sirtuin inhibition mechanisms are …

Are sirtuins viable targets for improving healthspan and lifespan?

JA Baur, Z Ungvari, RK Minor, DG Le Couteur… - Nature reviews Drug …, 2012 - nature.com
Although the increased lifespan of our populations illustrates the success of modern
medicine, the risk of develo** many diseases increases exponentially with old age …