In recent years, transition‐metal‐catalyzed C− H activation has become a key strategy in the
field of organic synthesis. Rhodium complexes are widely used as catalysts in a variety of …

Chiral sulfinyl compounds, sulfoxides, sulfoximines, sulfinamides, and other derivatives, play
an important role in asymmetric synthesis as versatile auxiliaries, ligands, and catalysts …

Sulfoximines have been largely disregarded in medicinal chemistry for a long time.
However, recently, they have risen to the apparent level of stardom on the drug discovery …

Chiral sulfur pharmacophores are crucial for drug discovery in bioscience and medicinal
chemistry. While the catalytic asymmetric synthesis of sulfoxides and sulfinate esters with …

sulfinamides, sulfonamides, and sulfonimidamides are in-demand motifs in medicinal
chemistry, yet methods for the synthesis of alkyl variants that start from simple, readily …

Historically, sulfoximines, sulfondiimines and sulfonimidamides have been neglected
pharmacophores in drug discovery even though they offer very interesting properties. This …

New methods for the general asymmetric synthesis of sulfonimidamides are of great interest
due to their applications in medicinal chemistry, agrochemical discovery, and academic …

Sulfur can form diverse S (IV) and S (VI) stereogenic centers, of which some have gained
significant attention recently due to their increasing use as pharmacophores in drug …

An increased interest to expand three-dimensional chemical space for the design of new
materials and medicines has created a demand for isosteric replacement groups of …

Sulfonamide derivatives are frequently seen structural motifs in medicinal chemistry. Almost
a century after Gerhard Domagk's pioneering work leading to the first sulfonamide antibiotic …