[HTML][HTML] ABCB1 and ABCG2 regulation at the blood-brain barrier: potential new targets to improve brain drug delivery

JA Schulz, AMS Hartz, B Bauer - Pharmacological Reviews, 2023‏ - Elsevier
The drug efflux transporters ABCB1 and ABCG2 at the blood-brain barrier limit the delivery
of drugs into the brain. Strategies to overcome ABCB1/ABCG2 have been largely …

ABC transporters at the blood–brain interfaces, their study models, and drug delivery implications in gliomas

D Gomez-Zepeda, M Taghi, JM Scherrmann… - Pharmaceutics, 2019‏ - mdpi.com
Drug delivery into the brain is regulated by the blood–brain interfaces. The blood–brain
barrier (BBB), the blood–cerebrospinal fluid barrier (BCSFB), and the blood–arachnoid …

Opioids and the blood-brain barrier: a dynamic interaction with consequences on drug disposition in brain

C Chaves, F Remiao, S Cisternino… - Current …, 2017‏ - benthamdirect.com
Background: Opioids are widely used in pain management, acting via opioid receptors
and/or Toll-like receptors (TLR) present at the central nervous system (CNS). At the blood …

The opioid epidemic: a central role for the blood brain barrier in opioid analgesia and abuse

CP Schaefer, ME Tome, TP Davis - Fluids and Barriers of the CNS, 2017‏ - Springer
Opioids are currently the primary treatment method used to manage both acute and chronic
pain. In the past two to three decades, there has been a surge in the use, abuse and misuse …

[HTML][HTML] Study models of drug–drug interactions involving p-glycoprotein: the potential benefit of p-glycoprotein modulation at the kidney and intestinal levels

J Veiga-Matos, AI Morales, M Prieto, F Remião, R Silva - Molecules, 2023‏ - mdpi.com
P-glycoprotein (P-gp) is a crucial membrane transporter situated on the cell's apical surface,
being responsible for eliminating xenobiotics and endobiotics. P-gp modulators are …

[HTML][HTML] The impact of P-glycoprotein on opioid analgesics: what's the real meaning in pain management and palliative care?

F Coluzzi, MS Scerpa, M Rocco… - International Journal of …, 2022‏ - mdpi.com
Opioids are widely used in cancer and non-cancer pain management. However, many
transporters at the blood–brain barrier (BBB), such as P-glycoprotein (P-gp, ABCB1/MDR1) …

Opioid and neuroHIV comorbidity–current and future perspectives

S Fitting, MP McRae, KF Hauser - Journal of Neuroimmune Pharmacology, 2020‏ - Springer
With the current national opioid crisis, it is critical to examine the mechanisms underlying
pathophysiologic interactions between human immunodeficiency virus (HIV) and opioids in …

[HTML][HTML] An interspecies molecular and functional study of organic cation transporters at the blood-brain barrier: from rodents to humans

C Chaves, F Campanelli, H Chapy, D Gomez-Zepeda… - Pharmaceutics, 2020‏ - mdpi.com
Organic cation transporters (OCTs) participate in the handling of compounds in kidneys and
at the synaptic cleft. Their role at the blood-brain barrier (BBB) in brain drug delivery is still …

[HTML][HTML] High-dose acetaminophen alters the integrity of the blood–brain barrier and leads to increased CNS uptake of codeine in rats

J Yang, RD Betterton, EI Williams, JA Stanton… - Pharmaceutics, 2022‏ - mdpi.com
The consumption of acetaminophen (APAP) can induce neurological changes in human
subjects; however, effects of APAP on blood–brain barrier (BBB) integrity are unknown. BBB …

[HTML][HTML] Characterization of the blood–brain barrier integrity and the brain transport of SN-38 in an orthotopic xenograft rat model of diffuse intrinsic pontine glioma

C Chaves, X Declèves, M Taghi, MC Menet, J Lacombe… - Pharmaceutics, 2020‏ - mdpi.com
The blood–brain barrier (BBB) hinders the brain delivery of many anticancer drugs. In
pediatric patients, diffuse intrinsic pontine glioma (DIPG) represents the main cause of brain …