ChemistGA: a chemical synthesizable accessible molecular generation algorithm for real-world drug discovery

J Wang, X Wang, H Sun, M Wang, Y Zeng… - Journal of Medicinal …, 2022 - ACS Publications
Many deep learning (DL)-based molecular generative models have been proposed to
design novel molecules. These models may perform well on benchmarks, but they usually …

ChemSpaceAL: An efficient active learning methodology applied to protein-specific molecular generation

GW Kyro, A Morgunov, RI Brent, VS Batista - Biophysical Journal, 2024 - cell.com
The incredible capabilities of generative artificial intelligence models have inevitably led to
their application in the domain of drug discovery. It is therefore of tremendous interest to …

[HTML][HTML] Designing mechanosensitive molecules from molecular building blocks: A genetic algorithm-based approach

M Blaschke, F Pauly - The Journal of Chemical Physics, 2023 - pubs.aip.org
Single molecules can be used as miniaturized functional electronic components, when
contacted by macroscopic electrodes. Mechanosensitivity describes a change in …

Inverse design of copolymers including stoichiometry and chain architecture

G Vogel, JM Weber - Chemical Science, 2025 - pubs.rsc.org
The demand for innovative synthetic polymers with improved properties is high, but their
structural complexity and vast design space hinder rapid discovery. Machine learning …

Development of Deep Learning approaches to predict relationships between chemical structures and sweetness

J Capela, J Correia, V Pereira… - 2022 International Joint …, 2022 - ieeexplore.ieee.org
The non-caloric sweeteners market is catching up with the market of conventionally used
sugars due to the benefits of preventing obesity, tooth decay and other health problems …

A Generative Evolutionary Many-Objective Framework: A Case Study in Antimicrobial Agent Design

MMP Da Silva, JS Angelo, IA Guedes… - Proceedings of the …, 2024 - dl.acm.org
de novo drug design (dnDD) aims to generate novel molecules that meet several conflicting
objectives, positioning it as a quintessential many-objective optimization problem (MaOP) …

Molecule optimization via multi-objective evolutionary in implicit chemical space

X **a, Y Su, C Zheng, X Zeng - arxiv preprint arxiv:2212.08826, 2022 - arxiv.org
Machine learning methods have been used to accelerate the molecule optimization process.
However, efficient search for optimized molecules satisfying several properties with scarce …

AI Enabled Drug Design and Side Effect Prediction Powered by Multi-Objective Evolutionary Algorithms & Transformer Models

K Grantham - 2023 - dr.library.brocku.ca
Due to the large search space and conflicting objectives, drug design and discovery is a
difficult problem for which new machine learning (ML) approaches are required. Here, the …