Sparks of function by de novo protein design

AE Chu, T Lu, PS Huang - Nature biotechnology, 2024 - nature.com
Abstract Information in proteins flows from sequence to structure to function, with each step
causally driven by the preceding one. Protein design is founded on inverting this process …

A survey of generative AI for de novo drug design: new frontiers in molecule and protein generation

X Tang, H Dai, E Knight, F Wu, Y Li, T Li… - Briefings in …, 2024 - academic.oup.com
Artificial intelligence (AI)-driven methods can vastly improve the historically costly drug
design process, with various generative models already in widespread use. Generative …

Artificial intelligence for science in quantum, atomistic, and continuum systems

X Zhang, L Wang, J Helwig, Y Luo, C Fu, Y **e… - arxiv preprint arxiv …, 2023 - arxiv.org
Advances in artificial intelligence (AI) are fueling a new paradigm of discoveries in natural
sciences. Today, AI has started to advance natural sciences by improving, accelerating, and …

On the design fundamentals of diffusion models: A survey

Z Chang, GA Koulieris, HPH Shum - arxiv preprint arxiv:2306.04542, 2023 - arxiv.org
Diffusion models are generative models, which gradually add and remove noise to learn the
underlying distribution of training data for data generation. The components of diffusion …

Point cloud approach to generative modeling for galaxy surveys at the field level

C Cuesta-Lazaro, S Mishra-Sharma - Physical Review D, 2024 - APS
We introduce a diffusion-based generative model to describe the distribution of galaxies in
our Universe directly as a collection of points in 3D space (coordinates) optionally with …

[HTML][HTML] ProteinReDiff: Complex-based ligand-binding proteins redesign by equivariant diffusion-based generative models

VTD Nguyen, ND Nguyen, TS Hy - Structural Dynamics, 2024 - pubs.aip.org
Proteins, serving as the fundamental architects of biological processes, interact with ligands
to perform a myriad of functions essential for life. Designing functional ligand-binding …

[HTML][HTML] Structure-based protein and small molecule generation using EGNN and diffusion models: A comprehensive review

F Soleymani, E Paquet, HL Viktor… - Computational and …, 2024 - Elsevier
Recent breakthroughs in deep learning have revolutionized protein sequence and structure
prediction. These advancements are built on decades of protein design efforts, and are …

Neural graph generator: Feature-conditioned graph generation using latent diffusion models

I Evdaimon, G Nikolentzos, C Xypolopoulos… - arxiv preprint arxiv …, 2024 - arxiv.org
Graph generation has emerged as a crucial task in machine learning, with significant
challenges in generating graphs that accurately reflect specific properties. Existing methods …

Deep learning in template-free de novo biosynthetic pathway design of natural products

X **e, L Gui, B Qiao, G Wang, S Huang… - Briefings in …, 2024 - academic.oup.com
Natural products (NPs) are indispensable in drug development, particularly in combating
infections, cancer, and neurodegenerative diseases. However, their limited availability …

Transferable deep generative modeling of intrinsically disordered protein conformations

G Janson, M Feig - PLOS Computational Biology, 2024 - journals.plos.org
Intrinsically disordered proteins have dynamic structures through which they play key
biological roles. The elucidation of their conformational ensembles is a challenging problem …