Advancements in the development of multi-target directed ligands for the treatment of Alzheimer's disease

N Kumar, V Kumar, P Anand, V Kumar… - Bioorganic & Medicinal …, 2022‏ - Elsevier
Alzheimer's disease (AD) is a multifactorial irreversible neurological disorder which results
in cognitive impairment, loss of cholinergic neurons in synapses of the basal forebrain and …

Novel therapeutic strategies for dementia

R Cacabelos, C Torrellas, I Carrera… - CNS & Neurological …, 2016‏ - ingentaconnect.com
Dementia represents a major problem of health and disability, with a relevant economic
impact on our society. Despite important advances in pathogenesis, diagnosis and …

Novel conjugates of aminoadamantanes with carbazole derivatives as potential multitarget agents for AD treatment

SO Bachurin, EF Shevtsova, GF Makhaeva… - Scientific Reports, 2017‏ - nature.com
A new group of compounds, promising for the design of original multitarget therapeutic
agents for treating neurodegenerative diseases, based on conjugates of aminoadamantane …

Hydrazides and hydrazones: Robust scaffolds in neurological and neurodegenerative disorders

N Agrawal, R Mishra, S Pathak… - Letters in Organic …, 2023‏ - benthamdirect.com
Background: Hydrazides and hydrazones are found in a variety of bioactive compounds that
have a wide range of pharmacological applications. There have been significant …

Synthesis, biological assessment and molecular docking study of new sulfur-linked 1, 2, 4-triazole and 1, 2, 3-triazole hybrid derivatives as potential DNA gyrase …

M El-Naggar, K Hasan, M Khanfar… - … für Naturforschung B, 2024‏ - degruyter.com
A series of new pyridine-1, 2, 4-triazole-tagged 1, 2, 3-triazole hybrid molecules were
obtained. The new compounds were synthesized via click chemistry of 1, 2, 4-triazole-3 …

[HTML][HTML] Chalcone scaffolds exhibiting acetylcholinesterase enzyme inhibition: Mechanistic and computational investigations

YA Malik, TA Awad, M Abdalla, S Yagi, HA Alhazmi… - Molecules, 2022‏ - mdpi.com
This study was aimed to perform the mechanistic investigations of chalcone scaffold as
inhibitors of acetylcholinesterase (AChE) enzyme using molecular docking and molecular …

[HTML][HTML] Synthesis, characterization and biological evaluation of metal adamantyl 2-pyridylhydrazone complexes

IA Shehadi, FA Delmani, AM Jaber, H Hammad… - Molecules, 2020‏ - mdpi.com
Four new complexes derived from adamantly containing hydrazone (APH) ligand with Cu
(II)(1), Co (II)(2), Ni (II)(3) and Zn (II)(4), have been synthesized and characterized using …

Novel iodinated hydrazide-hydrazones and their analogues as acetyl-and butyrylcholinesterase Inhibitors

M Krátký, Š Štěpánková, M Brablíková… - Current Topics in …, 2020‏ - benthamdirect.com
Background: Hydrazide-hydrazones have been known as scaffold with various biological
activities including inhibition of acetyl-(AChE) and butyrylcholinesterase (BuChE) …

Design, synthesis and antimicrobial assessments of aminoacetylenic-piperazine nitroimidazole hybrid compounds

AJ Rasras, RA Al-Qawasmeh, M El-Naggar… - … für Naturforschung C, 2023‏ - degruyter.com
A new series of aminoacetylenic nitroimidazole piperazine hybrid compounds were
prepared via three-component reaction. Mannich-type reaction was utilized to couple the …