Coumarin–benzimidazole hybrids: A review of developments in medicinal chemistry

R Gondru, Y Li, J Banothu - European Journal of Medicinal Chemistry, 2022 - Elsevier
Coumarin and benzimidazole are privileged structures in medicinal chemistry and are
widely used in drug discovery and development due to their vast biological properties. The …

Benzimidazole-triazole hybrids as antimicrobial and antiviral agents: A systematic review

M Marinescu - Antibiotics, 2023 - mdpi.com
Bacterial infections have attracted the attention of researchers in recent decades, especially
due to the special problems they have faced, such as their increasing diversity and …

New drugs are not enough-drug repositioning in oncology: An update

RG Armando, DLM Gomez… - … Journal of Oncology, 2020 - spandidos-publications.com
Drug repositioning refers to the concept of discovering novel clinical benefits of drugs that
are already known for use treating other diseases. The advantages of this are that several …

The nano-based catalyst for the synthesis of benzimidazoles

RS Keri, V Adimule, P Kendrekar, BS Sasidhar - Topics in Catalysis, 2022 - Springer
The properties of benzimidazole and its derivatives have been studied over more than one
hundred years. The benzimidazole ring is an important pharmacophore in modern drug …

Copper-Catalyzed Construction of Benzo[4,5]imidazo[2,1-a]isoquinolines Using Calcium Carbide as a Solid Alkyne Source

H Liu, Z Li - Organic Letters, 2021 - ACS Publications
A method for the synthesis of benzo [4, 5] imidazo [2, 1-a] isoquinolines through
Sonogashira cross-coupling/nucleophilic addition tandem reactions using calcium carbide …

Antimicrobial peptides and cationic nanoparticles: a broad-spectrum weapon to fight multi-drug resistance not only in bacteria

GE Valenti, S Alfei, D Caviglia, C Domenicotti… - International journal of …, 2022 - mdpi.com
In the last few years, antibiotic resistance and, analogously, anticancer drug resistance have
increased considerably, becoming one of the main public health problems. For this reason, it …

Recent advances in the anticancer applications of benzimidazole derivatives

M Mavvaji, S Akkoc - ChemistrySelect, 2023 - Wiley Online Library
Cancer, one of the most deadly diseases worldwide, is still a crucial challenge to human
well‐being. Hence, the design and development of modern protocols to cure diverse kinds …

SAR investigation and optimization of benzimidazole-based derivatives as antimicrobial agents against Gram-negative bacteria

EME Dokla, NS Abutaleb, SN Milik, EAEA Kandil… - European Journal of …, 2023 - Elsevier
Antibiotic-resistant bacteria represent a serious threat to modern medicine and human life.
Only a minority of antibacterial agents are active against Gram-negative bacteria. Hence, the …

Efficient synthesis of 1, 2-disubstituted benzimidazoles catalyzed by phosphoric acid as a homogeneous catalyst under mild conditions and investigating their anti …

AM Bistgani, A Dehghani, L Moradi - RSC advances, 2023 - pubs.rsc.org
A green practical method for the efficient synthesis of 1-benzyl-2-phenyl-benzimidazole and
its derivatives using phosphoric acid as an eco-friendly homogeneous catalyst from the …

Synthesis, Antimicrobial and Antibiofilm Activities, and Molecular Docking Investigations of 2-(1H-Indol-3-yl)-1H-benzo[d]imidazole Derivatives

EY Mendogralo, LY Nesterova, ER Nasibullina… - Molecules, 2023 - mdpi.com
The treatment of many bacterial and fungal infections remains a problem due to increasing
antibiotic resistance and biofilm formation by pathogens. In the present article, a …